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Discovery of ML210-Based glutathione peroxidase 4 (GPX4) degrader inducing ferroptosis of human cancer cells.
Wang, Han; Wang, Chao; Li, Bingru; Zheng, Cangxin; Liu, Guoquan; Liu, Zhenming; Zhang, Liangren; Xu, Ping.
Afiliación
  • Wang H; Department of Medicinal Chemistry, School of Pharmaceutical Sciences, Peking University, Beijing, China.
  • Wang C; State Key Laboratory of Natural and Biomimetic Drugs, Department of Medicinal Chemistry, School of Pharmaceutical Sciences, Peking University, Beijing, China. Electronic address: wangchao@bjmu.edu.cn.
  • Li B; State Key Laboratory of Natural and Biomimetic Drugs, Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing, China.
  • Zheng C; Department of Medicinal Chemistry, School of Pharmaceutical Sciences, Peking University, Beijing, China.
  • Liu G; State Key Laboratory of Natural and Biomimetic Drugs, Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing, China.
  • Liu Z; State Key Laboratory of Natural and Biomimetic Drugs, Department of Medicinal Chemistry, School of Pharmaceutical Sciences, Peking University, Beijing, China.
  • Zhang L; State Key Laboratory of Natural and Biomimetic Drugs, Department of Medicinal Chemistry, School of Pharmaceutical Sciences, Peking University, Beijing, China.
  • Xu P; Department of Medicinal Chemistry, School of Pharmaceutical Sciences, Peking University, Beijing, China. Electronic address: pingxu@bjmu.edu.cn.
Eur J Med Chem ; 254: 115343, 2023 Jun 05.
Article en En | MEDLINE | ID: mdl-37087895

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Ferroptosis / Neoplasias Límite: Animals / Humans Idioma: En Revista: Eur J Med Chem Año: 2023 Tipo del documento: Article País de afiliación: China Pais de publicación: Francia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Ferroptosis / Neoplasias Límite: Animals / Humans Idioma: En Revista: Eur J Med Chem Año: 2023 Tipo del documento: Article País de afiliación: China Pais de publicación: Francia