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Structure-Based Development of Isoform-Selective Inhibitors of Casein Kinase 1ε vs Casein Kinase 1δ.
Choi, Jun Yong; Noguchi, Yoshihiko; Alburger, James M; Bayle, Simon; Chung, Eugene; Grant, Wayne; Chaikuad, Apirat; Knapp, Stefan; Duckett, Derek R; Roush, William R.
Afiliación
  • Choi JY; Department of Chemistry, The Scripps Research Institute, Scripps Florida, Jupiter, Florida 33458, United States.
  • Noguchi Y; Department of Chemistry and Biochemistry, Queens College, Queens, New York 11367, United States.
  • Alburger JM; Ph.D. Programs in Chemistry and Biochemistry, The Graduate Center of the City University of New York, New York, New York 10016, United States.
  • Bayle S; Department of Chemistry, The Scripps Research Institute, Scripps Florida, Jupiter, Florida 33458, United States.
  • Chung E; Department of Chemistry, The Scripps Research Institute, Scripps Florida, Jupiter, Florida 33458, United States.
  • Grant W; Department of Drug Discovery, Moffitt Cancer Center, Tampa, Florida 33612, United States.
  • Chaikuad A; Department of Chemistry and Biochemistry, Queens College, Queens, New York 11367, United States.
  • Knapp S; Department of Molecular Therapeutics, The Scripps Research Institute, Scripps Florida, Jupiter, Florida 33458, United States.
  • Duckett DR; Institute of Pharmaceutical Chemistry, Goethe University, Frankfurt am Main 60438, Germany.
  • Roush WR; Structural Genomics Consortium, BMLS, Goethe University, Frankfurt am Main 60438, Germany.
J Med Chem ; 66(11): 7162-7178, 2023 06 08.
Article en En | MEDLINE | ID: mdl-37204207

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Quinasa Idelta de la Caseína Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Quinasa Idelta de la Caseína Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos