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Molecular mechanism of EAG1 channel inhibition by imipramine binding to the PAS domain.
Wang, Ze-Jun; Ghorbani, Mahdi; Chen, Xi; Tiwari, Purushottam B; Klauda, Jeffery B; Brelidze, Tinatin I.
Afiliación
  • Wang ZJ; Department of Pharmacology and Physiology, Georgetown University Medical Center, Washington, District of Columbia, USA.
  • Ghorbani M; Department of Chemical and Biomolecular Engineering, University of Maryland, College Park, Maryland, USA.
  • Chen X; Department of Pharmacology and Physiology, Georgetown University Medical Center, Washington, District of Columbia, USA.
  • Tiwari PB; Department of Oncology, Georgetown University Medical Center, Washington, District of Columbia, USA.
  • Klauda JB; Department of Chemical and Biomolecular Engineering, University of Maryland, College Park, Maryland, USA; Institute for Physical Science and Technology and Biophysics Graduate Program, University of Maryland, College Park, Maryland, USA. Electronic address: jbklauda@umd.edu.
  • Brelidze TI; Department of Pharmacology and Physiology, Georgetown University Medical Center, Washington, District of Columbia, USA. Electronic address: tib5@georgetown.edu.
J Biol Chem ; 299(12): 105391, 2023 Dec.
Article en En | MEDLINE | ID: mdl-37898402

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Canales de Potasio Éter-A-Go-Go / Imipramina Límite: Animals Idioma: En Revista: J Biol Chem Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Canales de Potasio Éter-A-Go-Go / Imipramina Límite: Animals Idioma: En Revista: J Biol Chem Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos