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Virtual Fragment Screening Identification of a Quinoline-5,8-dicarboxylic Acid Derivative as a Selective JMJD3 Inhibitor.
Giordano, Assunta; Del Gaudio, Federica; Johansson, Catrine; Riccio, Raffaele; Oppermann, Udo; Di Micco, Simone.
Affiliation
  • Giordano A; Institute of Biomolecular Chemistry (ICB), Consiglio Nazionale delle Ricerche (CNR), Via Campi Flegrei 34, 80078, Pozzuoli (Napoli), Italy.
  • Del Gaudio F; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II, 132, 84084, Fisciano (Salerno), Italy.
  • Johansson C; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II, 132, 84084, Fisciano (Salerno), Italy.
  • Riccio R; PhD Program in Drug Discovery and Development, University of Salerno, Via Giovanni Paolo II, 132, 84084, Fisciano (Salerno), Italy.
  • Oppermann U; Farmaceutici Damor S.p.A, Via E. Scaglione 27, 80145, Naples, Italy.
  • Di Micco S; Botnar Research Centre, Oxford NIHR BRU, Oxford University, Oxford Centre for Translational Myeloma Research, Oxford, OX3 7LD, UK.
ChemMedChem ; 13(12): 1160-1164, 2018 06 20.
Article in En | MEDLINE | ID: mdl-29633584

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinolines / Dicarboxylic Acids / Enzyme Inhibitors / Jumonji Domain-Containing Histone Demethylases / Isoenzymes Type of study: Diagnostic_studies / Screening_studies Limits: Humans Language: En Journal: ChemMedChem Journal subject: FARMACOLOGIA / QUIMICA Year: 2018 Document type: Article Affiliation country:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinolines / Dicarboxylic Acids / Enzyme Inhibitors / Jumonji Domain-Containing Histone Demethylases / Isoenzymes Type of study: Diagnostic_studies / Screening_studies Limits: Humans Language: En Journal: ChemMedChem Journal subject: FARMACOLOGIA / QUIMICA Year: 2018 Document type: Article Affiliation country: