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Synthesis and biological evaluation of carboxamide and quinoline derivatives as P2X7R antagonists.
Shah, Qasim; Hussain, Zahid; Ahmad Khan, Bilal; Jacobson, Kenneth A; Iqbal, Jamshed.
Affiliation
  • Shah Q; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad 22060, Pakistan; Department of Pharmacy, COMSATS University Islamabad, Abbottabad Campus, Abbottabad 22060, Pakistan.
  • Hussain Z; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad 22060, Pakistan.
  • Ahmad Khan B; Department of Chemistry, University of Azad Jammu and Kashmir, Muzaffarabad 13100, Pakistan.
  • Jacobson KA; Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda MD 20892, USA. Electronic address: kennethj@niddk.nih.gov.
  • Iqbal J; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad 22060, Pakistan; Department of Pharmacy, COMSATS University Islamabad, Abbottabad Campus, Abbottabad 22060, Pakistan. Electronic address: drjamshed@cuiatd.edu.pk.
Bioorg Chem ; 140: 106796, 2023 11.
Article in En | MEDLINE | ID: mdl-37683539

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinolines / Astrocytoma / Purinergic P2X Receptor Antagonists / Hydroxyquinolines Type of study: Prognostic_studies Limits: Humans Language: En Journal: Bioorg Chem Year: 2023 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinolines / Astrocytoma / Purinergic P2X Receptor Antagonists / Hydroxyquinolines Type of study: Prognostic_studies Limits: Humans Language: En Journal: Bioorg Chem Year: 2023 Document type: Article Affiliation country: Country of publication: