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Discovery of Clinical Candidate GSK1842799 As a Selective S1P1 Receptor Agonist (Prodrug) for Multiple Sclerosis.
Deng, Hongfeng; Bernier, Sylvie G; Doyle, Elisabeth; Lorusso, Jeanine; Morgan, Barry A; Westlin, William F; Evindar, Ghotas.
Affiliation
  • Deng H; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.
  • Bernier SG; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.
  • Doyle E; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.
  • Lorusso J; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.
  • Morgan BA; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.
  • Westlin WF; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.
  • Evindar G; Department of Medicinal Chemistry and Department of Preclinical Research, Praecis Pharmaceuticals Incorporated , 830 Winter Street, Waltham, Massachusetts 02451, United States.
ACS Med Chem Lett ; 4(10): 942-7, 2013 Oct 10.
Article de En | MEDLINE | ID: mdl-24900589

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Langue: En Journal: ACS Med Chem Lett Année: 2013 Type de document: Article Pays d'affiliation: États-Unis d'Amérique

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Langue: En Journal: ACS Med Chem Lett Année: 2013 Type de document: Article Pays d'affiliation: États-Unis d'Amérique