Your browser doesn't support javascript.
loading
Synthesis and SAR study of potent and selective PI3Kδ inhibitors.
Bui, Minna; Hao, Xiaolin; Shin, Youngsook; Cardozo, Mario; He, Xiao; Henne, Kirk; Suchomel, Julia; McCarter, John; McGee, Lawrence R; San Miguel, Tisha; Medina, Julio C; Mohn, Deanna; Tran, Thuy; Wannberg, Sharon; Wong, Jamie; Wong, Simon; Zalameda, Leeanne; Metz, Daniela; Cushing, Timothy D.
Affiliation
  • Bui M; Department of Therapeutic Discovery, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • Hao X; Department of Therapeutic Discovery, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • Shin Y; Department of Therapeutic Discovery, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • Cardozo M; Department of Therapeutic Discovery, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • He X; Department of Therapeutic Discovery, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • Henne K; Department of Pharmacokinetics and Drug Metabolism, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • Suchomel J; Department of Therapeutic Discovery, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • McCarter J; Department of Therapeutic Discovery, Amgen Inc., One Amgen Center Drive, Thousand Oaks, CA 91320, United States.
  • McGee LR; Department of Therapeutic Discovery, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • San Miguel T; Department of Inflammation Research, Amgen Inc., One Amgen Center Drive, Thousand Oaks, CA 91320, United States.
  • Medina JC; Department of Therapeutic Discovery, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • Mohn D; Department of Inflammation Research, Amgen Inc., One Amgen Center Drive, Thousand Oaks, CA 91320, United States.
  • Tran T; Department of Pharmacokinetics and Drug Metabolism, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • Wannberg S; Department of Inflammation Research, Amgen Inc., One Amgen Center Drive, Thousand Oaks, CA 91320, United States.
  • Wong J; Department of Pharmacokinetics and Drug Metabolism, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • Wong S; Department of Pharmacokinetics and Drug Metabolism, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
  • Zalameda L; Department of Inflammation Research, Amgen Inc., One Amgen Center Drive, Thousand Oaks, CA 91320, United States.
  • Metz D; Department of Inflammation Research, Amgen Inc., One Amgen Center Drive, Thousand Oaks, CA 91320, United States.
  • Cushing TD; Department of Therapeutic Discovery, Amgen Inc., 1120 Veterans Boulevard, South San Francisco, CA 94080, United States.
Bioorg Med Chem Lett ; 25(5): 1104-9, 2015 Mar 01.
Article de En | MEDLINE | ID: mdl-25666823

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: Quinoléines / Inhibiteurs de protéines kinases / Phosphatidylinositol 3-kinases de classe I Limites: Animals / Humans / Male Langue: En Journal: Bioorg Med Chem Lett Sujet du journal: BIOQUIMICA / QUIMICA Année: 2015 Type de document: Article Pays d'affiliation: États-Unis d'Amérique Pays de publication: Royaume-Uni

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: Quinoléines / Inhibiteurs de protéines kinases / Phosphatidylinositol 3-kinases de classe I Limites: Animals / Humans / Male Langue: En Journal: Bioorg Med Chem Lett Sujet du journal: BIOQUIMICA / QUIMICA Année: 2015 Type de document: Article Pays d'affiliation: États-Unis d'Amérique Pays de publication: Royaume-Uni