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Structure-Based Design of Selective Janus Kinase 2 Imidazo[4,5-d]pyrrolo[2,3-b]pyridine Inhibitors.
Hart, Amy C; Schroeder, Gretchen M; Wan, Honghe; Grebinski, James; Inghrim, Jennifer; Kempson, James; Guo, Junqing; Pitts, William J; Tokarski, John S; Sack, John S; Khan, Javed A; Lippy, Jonathan; Lorenzi, Matthew V; You, Dan; McDevitt, Theresa; Vuppugalla, Ragini; Zhang, Yueping; Lombardo, Louis J; Trainor, George L; Purandare, Ashok V.
Affiliation
  • Hart AC; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Schroeder GM; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Wan H; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Grebinski J; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Inghrim J; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Kempson J; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Guo J; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Pitts WJ; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Tokarski JS; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Sack JS; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Khan JA; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Lippy J; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Lorenzi MV; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • You D; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • McDevitt T; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Vuppugalla R; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Zhang Y; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Lombardo LJ; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Trainor GL; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
  • Purandare AV; Bristol-Myers Squibb Research & Development , Princeton, New Jersey 08543, United States.
ACS Med Chem Lett ; 6(8): 845-9, 2015 Aug 13.
Article de En | MEDLINE | ID: mdl-26288682

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Langue: En Journal: ACS Med Chem Lett Année: 2015 Type de document: Article Pays d'affiliation: États-Unis d'Amérique Pays de publication: États-Unis d'Amérique

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Langue: En Journal: ACS Med Chem Lett Année: 2015 Type de document: Article Pays d'affiliation: États-Unis d'Amérique Pays de publication: États-Unis d'Amérique