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Identification of flavonolignans from Silybum marianum seeds as allosteric protein tyrosine phosphatase 1B inhibitors.
Qin, Ningbo; Sasaki, Tatsunori; Li, Wei; Wang, Jian; Zhang, Xiangyu; Li, Dahong; Li, Zhanlin; Cheng, Maosheng; Hua, Huiming; Koike, Kazuo.
Affiliation
  • Qin N; a Key Laboratory of Structure-Based Drug Design & Discovery, Ministry of Education , Shenyang Pharmaceutical University , Shenyang , Liaoning , PR China.
  • Sasaki T; b School of Traditional Chinese Materia Medica , Shenyang Pharmaceutical University , Shenyang , Liaoning PR China.
  • Li W; c Faculty of Pharmaceutical Sciences , Toho University , Funabashi , Japan.
  • Wang J; a Key Laboratory of Structure-Based Drug Design & Discovery, Ministry of Education , Shenyang Pharmaceutical University , Shenyang , Liaoning , PR China.
  • Zhang X; c Faculty of Pharmaceutical Sciences , Toho University , Funabashi , Japan.
  • Li D; a Key Laboratory of Structure-Based Drug Design & Discovery, Ministry of Education , Shenyang Pharmaceutical University , Shenyang , Liaoning , PR China.
  • Li Z; d School of Pharmaceutical Engineering , Shenyang Pharmaceutical University , Shenyang , Liaoning , PR China.
  • Cheng M; a Key Laboratory of Structure-Based Drug Design & Discovery, Ministry of Education , Shenyang Pharmaceutical University , Shenyang , Liaoning , PR China.
  • Hua H; d School of Pharmaceutical Engineering , Shenyang Pharmaceutical University , Shenyang , Liaoning , PR China.
  • Koike K; a Key Laboratory of Structure-Based Drug Design & Discovery, Ministry of Education , Shenyang Pharmaceutical University , Shenyang , Liaoning , PR China.
J Enzyme Inhib Med Chem ; 33(1): 1283-1291, 2018 Dec.
Article de En | MEDLINE | ID: mdl-30160205

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: Graines / Asteraceae / Flavonolignanes / Antienzymes / Protein Tyrosine Phosphatase, Non-Receptor Type 1 Type d'étude: Diagnostic_studies Limites: Humans Langue: En Journal: J Enzyme Inhib Med Chem Sujet du journal: BIOQUIMICA / QUIMICA Année: 2018 Type de document: Article

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: Graines / Asteraceae / Flavonolignanes / Antienzymes / Protein Tyrosine Phosphatase, Non-Receptor Type 1 Type d'étude: Diagnostic_studies Limites: Humans Langue: En Journal: J Enzyme Inhib Med Chem Sujet du journal: BIOQUIMICA / QUIMICA Année: 2018 Type de document: Article