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Discovery of Novel pERK1/2- or ß-Arrestin-Preferring 5-HT1A Receptor-Biased Agonists: Diversified Therapeutic-like versus Side Effect Profile.
Sniecikowska, Joanna; Gluch-Lutwin, Monika; Bucki, Adam; Wieckowska, Anna; Siwek, Agata; Jastrzebska-Wiesek, Magdalena; Partyka, Anna; Wilczynska, Daria; Pytka, Karolina; Latacz, Gniewomir; Przejczowska-Pomierny, Katarzyna; Wyska, Elzbieta; Wesolowska, Anna; Pawlowski, Maciej; Newman-Tancredi, Adrian; Kolaczkowski, Marcin.
Affiliation
  • Sniecikowska J; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Gluch-Lutwin M; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Bucki A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Wieckowska A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Siwek A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Jastrzebska-Wiesek M; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Partyka A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Wilczynska D; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Pytka K; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Latacz G; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Przejczowska-Pomierny K; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Wyska E; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Wesolowska A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Pawlowski M; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
  • Newman-Tancredi A; Neurolixis, Castres, France.
  • Kolaczkowski M; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
J Med Chem ; 63(19): 10946-10971, 2020 10 08.
Article de En | MEDLINE | ID: mdl-32883072

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: Conception de médicament / Agonistes des récepteurs de la sérotonine / Système de signalisation des MAP kinases / Bêta-Arrestines Type d'étude: Prognostic_studies Limites: Animals Langue: En Journal: J Med Chem Sujet du journal: QUIMICA Année: 2020 Type de document: Article Pays d'affiliation: Pologne Pays de publication: États-Unis d'Amérique

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: Conception de médicament / Agonistes des récepteurs de la sérotonine / Système de signalisation des MAP kinases / Bêta-Arrestines Type d'étude: Prognostic_studies Limites: Animals Langue: En Journal: J Med Chem Sujet du journal: QUIMICA Année: 2020 Type de document: Article Pays d'affiliation: Pologne Pays de publication: États-Unis d'Amérique