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Structure-activity relationship studies on divalent naphthalene diimide G quadruplex ligands with anticancer and antiparasitic activity.
Pérez-Soto, Manuel; Peñalver, Pablo; Street, Steven T G; Weenink, Dora; O'Hagan, Michael P; Ramos-Soriano, Javier; Jiang, Y Jennifer; Hollingworth, Gregory J; Galan, M Carmen; Morales, Juan C.
Affiliation
  • Pérez-Soto M; Instituto de Parasitología y Biomedicina, Avenida del Conocimiento, s/n 18016, Armilla, Granada, Spain.
  • Peñalver P; Instituto de Parasitología y Biomedicina, Avenida del Conocimiento, s/n 18016, Armilla, Granada, Spain.
  • Street STG; School of Chemistry, University of Bristol, Bristol BS8 1TS, United Kingdom.
  • Weenink D; Instituto de Parasitología y Biomedicina, Avenida del Conocimiento, s/n 18016, Armilla, Granada, Spain.
  • O'Hagan MP; School of Chemistry, University of Bristol, Bristol BS8 1TS, United Kingdom.
  • Ramos-Soriano J; School of Chemistry, University of Bristol, Bristol BS8 1TS, United Kingdom.
  • Jiang YJ; School of Chemistry, University of Bristol, Bristol BS8 1TS, United Kingdom.
  • Hollingworth GJ; Novartis Institutes for Biomedical Research, Novartis Campus, CH-4002 Basel, Switzerland.
  • Galan MC; School of Chemistry, University of Bristol, Bristol BS8 1TS, United Kingdom. Electronic address: M.C.Galan@bristol.ac.uk.
  • Morales JC; Instituto de Parasitología y Biomedicina, Avenida del Conocimiento, s/n 18016, Armilla, Granada, Spain. Electronic address: jcmorales@ipb.csic.es.
Bioorg Med Chem ; 71: 116946, 2022 10 01.
Article de En | MEDLINE | ID: mdl-35939903

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: G-quadruplexes / Antiparasitaires Langue: En Journal: Bioorg Med Chem Sujet du journal: BIOQUIMICA / QUIMICA Année: 2022 Type de document: Article Pays d'affiliation: Espagne Pays de publication: Royaume-Uni

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: G-quadruplexes / Antiparasitaires Langue: En Journal: Bioorg Med Chem Sujet du journal: BIOQUIMICA / QUIMICA Année: 2022 Type de document: Article Pays d'affiliation: Espagne Pays de publication: Royaume-Uni