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Neurotensin Receptor Allosterism Revealed in Complex with a Biased Allosteric Modulator.
Krumm, Brian E; DiBerto, Jeffrey F; Olsen, Reid H J; Kang, Hye Jin; Slocum, Samuel T; Zhang, Shicheng; Strachan, Ryan T; Huang, Xi-Ping; Slosky, Lauren M; Pinkerton, Anthony B; Barak, Lawrence S; Caron, Marc G; Kenakin, Terry; Fay, Jonathan F; Roth, Bryan L.
Affiliation
  • Krumm BE; Department of Pharmacology, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • DiBerto JF; Department of Pharmacology, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • Olsen RHJ; Department of Pharmacology, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • Kang HJ; Department of Pharmacology, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • Slocum ST; National Institute of Mental Health Psychoactive Drug Screening Program (NIMH PDSP), School of Medicine, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • Zhang S; Department of Pharmacology, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • Strachan RT; National Institute of Mental Health Psychoactive Drug Screening Program (NIMH PDSP), School of Medicine, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • Huang XP; Department of Pharmacology, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • Slosky LM; Department of Pharmacology, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • Pinkerton AB; Department of Pharmacology, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • Barak LS; National Institute of Mental Health Psychoactive Drug Screening Program (NIMH PDSP), School of Medicine, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599-7365, United States.
  • Caron MG; Department of Pharmacology, University of Minnesota, Minneapolis, Minnesota 55455, United States.
  • Kenakin T; Conrad Prebys Center for Chemical Genomics at Sanford Burnham Prebys Medical Discovery Institute, La Jolla, California 92037, United States.
  • Fay JF; Department of Cell Biology, Duke University, Durham, North Carolina 27710, United States.
  • Roth BL; Department of Cell Biology, Duke University, Durham, North Carolina 27710, United States.
Biochemistry ; 62(7): 1233-1248, 2023 04 04.
Article de En | MEDLINE | ID: mdl-36917754

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: Neurotensine / Récepteur neurotensine Langue: En Journal: Biochemistry Année: 2023 Type de document: Article Pays d'affiliation: États-Unis d'Amérique Pays de publication: États-Unis d'Amérique

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: Neurotensine / Récepteur neurotensine Langue: En Journal: Biochemistry Année: 2023 Type de document: Article Pays d'affiliation: États-Unis d'Amérique Pays de publication: États-Unis d'Amérique