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Discovery of novel triazine derivatives as potent retinoic acid receptor-related orphan receptor γt (RORγt) inverse agonists.
Lu, Lixue; Chen, Song; Yu, Mingcheng; Zhou, Ronghui; Guo, Siqi; Chen, Ji-An; Wang, Haojie; Chen, Shijie; Luo, Cheng; Xie, Qiong; Wang, Yonghui.
Affiliation
  • Lu L; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai, 201203, China.
  • Chen S; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai, 201203, China.
  • Yu M; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai, 201203, China.
  • Zhou R; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai, 201203, China.
  • Guo S; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai, 201203, China.
  • Chen JA; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai, 201203, China.
  • Wang H; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai, 201203, China.
  • Chen S; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai, 201203, China.
  • Luo C; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai, 201203, China.
  • Xie Q; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai, 201203, China; Fudan Zhangjiang Institute, Shanghai, 201203, China. Electronic address: qxie@fudan.edu.cn.
  • Wang Y; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai, 201203, China. Electronic address: yonghuiwang@fudan.edu.cn.
Eur J Med Chem ; 256: 115424, 2023 Aug 05.
Article de En | MEDLINE | ID: mdl-37167779

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: Maladies auto-immunes / Récepteurs à l'acide rétinoïque Limites: Animals Langue: En Journal: Eur J Med Chem Année: 2023 Type de document: Article Pays d'affiliation: Chine Pays de publication: France

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Sujet principal: Maladies auto-immunes / Récepteurs à l'acide rétinoïque Limites: Animals Langue: En Journal: Eur J Med Chem Année: 2023 Type de document: Article Pays d'affiliation: Chine Pays de publication: France