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3D-Shaped Binders of Unfolded Proteins Inducing Cancer Cell-Specific Endoplasmic Reticulum Stress In Vitro and In Vivo.
Klemt, Insa; Varzatskii, Oleg; Selin, Roman; Vakarov, Serhii; Kovalska, Vladyslava; Bila, Galyna; Bilyy, Rostyslav; Voloshin, Yan; Cuartero, Itziar Cossío; Hidalgo, Andrés; Frey, Benjamin; Becker, Ina; Friedrich, Bernhard; Tietze, Rainer; Friedrich, Ralf P; Alexiou, Christoph; Ursu, Elena-Laura; Rotaru, Alexandru; Solymosi, Iris; Pérez-Ojeda, M Eugenia; Mokhir, Andriy.
Affiliation
  • Klemt I; Department of Chemistry and Pharmacy, Organic Chemistry II, Friedrich-Alexander-University of Erlangen-Nürnberg (FAU), 91058 Erlangen, Germany.
  • Varzatskii O; Princeton Biomolecular Research Laboratories, 26A Saperne Pole Street, 01042 Kyiv, Ukraine.
  • Selin R; V.I. Vernadsky Institute of General and Inorganic Chemistry, NASU, 32/34 Palladin Av., 03142 Kyiv, Ukraine.
  • Vakarov S; Department of Chemistry and Pharmacy, Organic Chemistry II, Friedrich-Alexander-University of Erlangen-Nürnberg (FAU), 91058 Erlangen, Germany.
  • Kovalska V; Princeton Biomolecular Research Laboratories, 26A Saperne Pole Street, 01042 Kyiv, Ukraine.
  • Bila G; V.I. Vernadsky Institute of General and Inorganic Chemistry, NASU, 32/34 Palladin Av., 03142 Kyiv, Ukraine.
  • Bilyy R; Princeton Biomolecular Research Laboratories, 26A Saperne Pole Street, 01042 Kyiv, Ukraine.
  • Voloshin Y; Institute of Molecular Biology and Genetics, NASU, 150 Zabolotnogo Street, 03143 Kyiv, Ukraine.
  • Cuartero IC; Department of Histology, Cytology and Embryology, Danylo Halytsky Lviv National Medical University, Pekarska Street 69, 79010 Lviv, Ukraine.
  • Hidalgo A; Lectinotest R&D, Mechanichna Street 2, 79024 Lviv, Ukraine.
  • Frey B; Department of Histology, Cytology and Embryology, Danylo Halytsky Lviv National Medical University, Pekarska Street 69, 79010 Lviv, Ukraine.
  • Becker I; Lectinotest R&D, Mechanichna Street 2, 79024 Lviv, Ukraine.
  • Friedrich B; Nesmeyanov Institute of Organoelement Compounds, RAS, 28 Vavilova Street, 119334 Moscow, Russia.
  • Tietze R; Program of Cardiovascular Regeneration, Centro Nacional de Investigaciones Cardiovasculares Carlos III (CNIC), C. Melchor Fernández Almagro, 3, 28029 Madrid, Spain.
  • Friedrich RP; Program of Cardiovascular Regeneration, Centro Nacional de Investigaciones Cardiovasculares Carlos III (CNIC), C. Melchor Fernández Almagro, 3, 28029 Madrid, Spain.
  • Alexiou C; Department of Radiation Oncology, Translational Radiobiology, Universitaetsklinikum Erlangen, Friedrich-Alexander-University of Erlangen-Nürnberg (FAU), Glueckstrasse 4A, 91054 Erlangen, Germany.
  • Ursu EL; Department of Radiation Oncology, Translational Radiobiology, Universitaetsklinikum Erlangen, Friedrich-Alexander-University of Erlangen-Nürnberg (FAU), Glueckstrasse 4A, 91054 Erlangen, Germany.
  • Rotaru A; Department of Otorhinolaryngology, Head and Neck Surgery, Section of Experimental Oncology and Nanomedicine (SEON), University Hospital, Friedrich-Alexander-University of Erlangen-Nürnberg (FAU), Glückstraße 10a, 91054 Erlangen, Germany.
  • Solymosi I; Department of Otorhinolaryngology, Head and Neck Surgery, Section of Experimental Oncology and Nanomedicine (SEON), University Hospital, Friedrich-Alexander-University of Erlangen-Nürnberg (FAU), Glückstraße 10a, 91054 Erlangen, Germany.
  • Pérez-Ojeda ME; Department of Otorhinolaryngology, Head and Neck Surgery, Section of Experimental Oncology and Nanomedicine (SEON), University Hospital, Friedrich-Alexander-University of Erlangen-Nürnberg (FAU), Glückstraße 10a, 91054 Erlangen, Germany.
  • Mokhir A; Department of Otorhinolaryngology, Head and Neck Surgery, Section of Experimental Oncology and Nanomedicine (SEON), University Hospital, Friedrich-Alexander-University of Erlangen-Nürnberg (FAU), Glückstraße 10a, 91054 Erlangen, Germany.
J Am Chem Soc ; 145(40): 22252-22264, 2023 Oct 11.
Article de En | MEDLINE | ID: mdl-37773090

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Langue: En Journal: J Am Chem Soc Année: 2023 Type de document: Article Pays d'affiliation: Allemagne Pays de publication: États-Unis d'Amérique

Texte intégral: 1 Collection: 01-internacional Base de données: MEDLINE Langue: En Journal: J Am Chem Soc Année: 2023 Type de document: Article Pays d'affiliation: Allemagne Pays de publication: États-Unis d'Amérique