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Structure-based design of TACE selective inhibitors: manipulations in the S1'-S3' pocket.
Huang, Adrian; Joseph-McCarthy, Diane; Lovering, Frank; Sun, Linhong; Wang, Weiheng; Xu, Weixin; Zhu, Yi; Cui, Junqing; Zhang, Yuhua; Levin, Jeremy I.
Affiliation
  • Huang A; Chemical and Screening Sciences, Wyeth Research, 200 CambridgePark Drive, Cambridge, MA 02140, USA. ahuang@wyeth.com
Bioorg Med Chem ; 15(18): 6170-81, 2007 Sep 15.
Article in En | MEDLINE | ID: mdl-17606376
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Collection: 01-internacional Database: MEDLINE Main subject: Enzyme Inhibitors / ADAM Proteins / Hydroxamic Acids Type of study: Prognostic_studies Limits: Animals Language: En Journal: Bioorg Med Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2007 Document type: Article Affiliation country: Country of publication:
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Collection: 01-internacional Database: MEDLINE Main subject: Enzyme Inhibitors / ADAM Proteins / Hydroxamic Acids Type of study: Prognostic_studies Limits: Animals Language: En Journal: Bioorg Med Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2007 Document type: Article Affiliation country: Country of publication: