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Synthesis and activity of quinolinylmethyl P1' alpha-sulfone piperidine hydroxamate inhibitors of TACE.
Zhang, Chunchun; Lovering, Frank; Behnke, Mark; Zask, Arie; Sandanayaka, Vincent; Sun, Linhong; Zhu, Yi; Xu, Weixin; Zhang, Yuhua; Levin, Jeremy I.
Affiliation
  • Zhang C; Chemical and Screening Science, Wyeth Research, 401 N. Middletown Road, Pearl River, NY 10965, USA. zhangc9@wyeth.com
Bioorg Med Chem Lett ; 19(13): 3445-8, 2009 Jul 01.
Article in En | MEDLINE | ID: mdl-19464885

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperidines / Protease Inhibitors / Sulfones / ADAM Proteins / Hydroxamic Acids Limits: Animals / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2009 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperidines / Protease Inhibitors / Sulfones / ADAM Proteins / Hydroxamic Acids Limits: Animals / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2009 Document type: Article Affiliation country: Country of publication: