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Synthesis and evaluation of carbamoylmethylene linked prodrugs of BMS-582949, a clinical p38α inhibitor.
Liu, Chunjian; Lin, James; Everlof, Gerry; Gesenberg, Christoph; Zhang, Hongjian; Marathe, Punit H; Malley, Mary; Galella, Michael A; McKinnon, Murray; Dodd, John H; Barrish, Joel C; Schieven, Gary L; Leftheris, Katerina.
Affiliation
  • Liu C; Bristol-Myers Squibb Research and Development, PO Box 4000, Princeton, NJ 08543-4000, United States. chunjian.liu@bms.com
Bioorg Med Chem Lett ; 23(10): 3028-33, 2013 May 15.
Article in En | MEDLINE | ID: mdl-23578688

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyrroles / Triazines / Prodrugs / Dacarbazine / P38 Mitogen-Activated Protein Kinases / Protein Kinase Inhibitors Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2013 Document type: Article Affiliation country:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyrroles / Triazines / Prodrugs / Dacarbazine / P38 Mitogen-Activated Protein Kinases / Protein Kinase Inhibitors Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2013 Document type: Article Affiliation country: