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6-Phenylpyrimidin-4-ones as Positive Allosteric Modulators at the M1 mAChR: The Determinants of Allosteric Activity.
Jörg, Manuela; van der Westhuizen, Emma T; Khajehali, Elham; Burger, Wessel A C; White, Jonathan M; Choy, Kwok H C; Tobin, Andrew B; Sexton, Patrick M; Valant, Celine; Capuano, Ben; Christopoulos, Arthur; Scammells, Peter J.
Affiliation
  • White JM; Bio21 Molecular Science and Biotechnology Institute , The University of Melbourne , 30 Flemington Road , Parkville 3010 , VIC , Australia.
  • Tobin AB; Centre for Translational Pharmacology, Institute of Molecular, Cell and Systems Biology, College of Medical, Veterinary and Life Sciences , University of Glasgow , Glasgow G12 8QQ , United Kingdom.
ACS Chem Neurosci ; 10(3): 1099-1114, 2019 03 20.
Article in En | MEDLINE | ID: mdl-30547573

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyrimidines / Quinolines / Receptor, Muscarinic M1 Limits: Animals Language: En Journal: ACS Chem Neurosci Year: 2019 Document type: Article Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyrimidines / Quinolines / Receptor, Muscarinic M1 Limits: Animals Language: En Journal: ACS Chem Neurosci Year: 2019 Document type: Article Country of publication: