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CDK8 as a therapeutic target for cancers and recent developments in discovery of CDK8 inhibitors.
Xi, Meiyang; Chen, Tingkai; Wu, Chunlei; Gao, Xiaozhong; Wu, Yonghua; Luo, Xiang; Du, Kui; Yu, Lemao; Cai, Tao; Shen, Runpu; Sun, Haopeng.
Affiliation
  • Xi M; College of Chemistry and Chemical Engineering, Shaoxing University, Shaoxing, 312000, China.
  • Chen T; Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 210009, China.
  • Wu C; College of Chemistry and Chemical Engineering, Shaoxing University, Shaoxing, 312000, China.
  • Gao X; College of Chemistry and Chemical Engineering, Shaoxing University, Shaoxing, 312000, China.
  • Wu Y; College of Chemistry and Chemical Engineering, Shaoxing University, Shaoxing, 312000, China.
  • Luo X; College of Chemistry and Chemical Engineering, Shaoxing University, Shaoxing, 312000, China.
  • Du K; College of Chemistry and Chemical Engineering, Shaoxing University, Shaoxing, 312000, China.
  • Yu L; College of Chemistry and Chemical Engineering, Shaoxing University, Shaoxing, 312000, China.
  • Cai T; College of Chemistry and Chemical Engineering, Shaoxing University, Shaoxing, 312000, China.
  • Shen R; College of Chemistry and Chemical Engineering, Shaoxing University, Shaoxing, 312000, China.
  • Sun H; Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 210009, China. Electronic address: sunhaopeng@163.com.
Eur J Med Chem ; 164: 77-91, 2019 Feb 15.
Article in En | MEDLINE | ID: mdl-30594029

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protein Kinase Inhibitors / Cyclin-Dependent Kinase 8 / Neoplasms Limits: Humans Language: En Journal: Eur J Med Chem Year: 2019 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protein Kinase Inhibitors / Cyclin-Dependent Kinase 8 / Neoplasms Limits: Humans Language: En Journal: Eur J Med Chem Year: 2019 Document type: Article Affiliation country: Country of publication: