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Divinylsulfonamides enable the construction of homogeneous antibody-drug conjugates.
Huang, Rong; Sheng, Yao; Wei, Ding; Lu, Wenwen; Xu, Zili; Chen, Hongli; Jiang, Biao.
Affiliation
  • Huang R; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China; University of Chinese Academy of Sciences, 19A Yuquan Road, Shijingshan District, Beijing 100049, China.
  • Sheng Y; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China.
  • Wei D; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China; University of Chinese Academy of Sciences, 19A Yuquan Road, Shijingshan District, Beijing 100049, China; Shanghai Advanced Research Institute, Chinese Academy of S
  • Lu W; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China; University of Chinese Academy of Sciences, 19A Yuquan Road, Shijingshan District, Beijing 100049, China.
  • Xu Z; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China; University of Chinese Academy of Sciences, 19A Yuquan Road, Shijingshan District, Beijing 100049, China.
  • Chen H; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China. Electronic address: chenhl@shanghaitech.edu.cn.
  • Jiang B; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China. Electronic address: jiangbiao@shanghaitech.edu.cn.
Bioorg Med Chem ; 28(23): 115793, 2020 12 01.
Article in En | MEDLINE | ID: mdl-33039798

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Sulfonamides / Immunoconjugates Limits: Animals / Humans / Male Language: En Journal: Bioorg Med Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2020 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Sulfonamides / Immunoconjugates Limits: Animals / Humans / Male Language: En Journal: Bioorg Med Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2020 Document type: Article Affiliation country: Country of publication: