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Small-molecule inhibitors targeting Polycomb repressive complex 1 RING domain.
Shukla, Shirish; Ying, Weijiang; Gray, Felicia; Yao, Yiwu; Simes, Miranda L; Zhao, Qingjie; Miao, Hongzhi; Cho, Hyo Je; González-Alonso, Paula; Winkler, Alyssa; Lund, George; Purohit, Trupta; Kim, EunGi; Zhang, Xiaotian; Ray, Joshua M; He, Shihan; Nikolaidis, Caroline; Ndoj, Juliano; Wang, Jingya; Jaremko, Lukasz; Jaremko, Mariusz; Ryan, Russell J H; Guzman, Monica L; Grembecka, Jolanta; Cierpicki, Tomasz.
Affiliation
  • Shukla S; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Ying W; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Gray F; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Yao Y; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Simes ML; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Zhao Q; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Miao H; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Cho HJ; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • González-Alonso P; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Winkler A; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Lund G; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Purohit T; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Kim E; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Zhang X; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Ray JM; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • He S; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Nikolaidis C; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Ndoj J; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Wang J; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Jaremko L; MedImmune, LLC, Gaithersburg, MD, USA.
  • Jaremko M; Biological and Environmental Science and Engineering (BESE), King Abdullah University of Science and Technology (KAUST), Thuwal, Saudi Arabia.
  • Ryan RJH; Biological and Environmental Science and Engineering (BESE), King Abdullah University of Science and Technology (KAUST), Thuwal, Saudi Arabia.
  • Guzman ML; Department of Pathology, University of Michigan, Ann Arbor, MI, USA.
  • Grembecka J; Division of Hematology and Medical Oncology, Leukemia Program, Weill Cornell Medicine/New York-Presbyterian Hospital, New York, NY, USA.
  • Cierpicki T; Department of Pathology, University of Michigan, Ann Arbor, MI, USA. jolantag@umich.edu.
Nat Chem Biol ; 17(7): 784-793, 2021 07.
Article in En | MEDLINE | ID: mdl-34155404

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Small Molecule Libraries / Polycomb Repressive Complex 1 Limits: Humans Language: En Journal: Nat Chem Biol Journal subject: BIOLOGIA / QUIMICA Year: 2021 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Small Molecule Libraries / Polycomb Repressive Complex 1 Limits: Humans Language: En Journal: Nat Chem Biol Journal subject: BIOLOGIA / QUIMICA Year: 2021 Document type: Article Affiliation country: Country of publication: