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A multi-pronged evaluation of aldehyde-based tripeptidyl main protease inhibitors as SARS-CoV-2 antivirals.
Ma, Yuying; Yang, Kai S; Geng, Zhi Zachary; Alugubelli, Yugendar R; Shaabani, Namir; Vatansever, Erol C; Ma, Xinyu R; Cho, Chia-Chuan; Khatua, Kaustav; Xiao, Jing; Blankenship, Lauren R; Yu, Ge; Sankaran, Banumathi; Li, Pingwei; Allen, Robert; Ji, Henry; Xu, Shiqing; Liu, Wenshe Ray.
Affiliation
  • Ma Y; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Yang KS; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Geng ZZ; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Alugubelli YR; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Shaabani N; Sorrento Therapeutics, Inc. San Diego, CA, 92121, USA.
  • Vatansever EC; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Ma XR; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Cho CC; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Khatua K; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Xiao J; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Blankenship LR; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Yu G; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA.
  • Sankaran B; Molecular Biophysics and Integrated Bioimaging, Berkeley Center for Structural Biology, Laurence Berkeley National Laboratory, Berkeley, CA, 94720, USA.
  • Li P; Department of Biochemistry and Biophysics, Texas A&M University, College Station, TX, 77843, USA.
  • Allen R; Sorrento Therapeutics, Inc. San Diego, CA, 92121, USA.
  • Ji H; Sorrento Therapeutics, Inc. San Diego, CA, 92121, USA. Electronic address: hji@sorrentotherapeutics.com.
  • Xu S; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA. Electronic address: shiqing.xu@tamu.edu.
  • Liu WR; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, TX, 77843, USA; Department of Biochemistry and Biophysics, Texas A&M University, College Station, TX, 77843, USA; Institute of Biosciences and Technology and Department of Translational M
Eur J Med Chem ; 240: 114570, 2022 Oct 05.
Article in En | MEDLINE | ID: mdl-35779291

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: SARS-CoV-2 / COVID-19 Limits: Humans Language: En Journal: Eur J Med Chem Year: 2022 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: SARS-CoV-2 / COVID-19 Limits: Humans Language: En Journal: Eur J Med Chem Year: 2022 Document type: Article Affiliation country: Country of publication: