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Dopamine D3/D2 Receptor Antagonist PF-4363467 Attenuates Opioid Drug-Seeking Behavior without Concomitant D2 Side Effects.
Wager, Travis T; Chappie, Thomas; Horton, David; Chandrasekaran, Ramalakshmi Y; Samas, Brian; Dunn-Sims, Elizabeth R; Hsu, Cathleen; Nawreen, Nawshaba; Vanase-Frawley, Michelle A; O'Connor, Rebecca E; Schmidt, Christopher J; Dlugolenski, Keith; Stratman, Nancy C; Majchrzak, Mark J; Kormos, Bethany L; Nguyen, David P; Sawant-Basak, Aarti; Mead, Andy N.
Afiliação
  • Wager TT; Pfizer Worldwide Research and Development , Neuroscience Medicinal Chemistry and Neuroscience Research Unit, 610 Main Street, Cambridge, Massachusetts 02139, United States.
  • Chappie T; Pfizer Worldwide Research and Development , Neuroscience Medicinal Chemistry and Neuroscience Research Unit, 610 Main Street, Cambridge, Massachusetts 02139, United States.
  • Horton D; Pfizer Worldwide Research and Development , Chemistry and Biology, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Chandrasekaran RY; Pfizer Worldwide Research and Development , Chemistry and Biology, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Samas B; Pfizer Worldwide Research and Development , Chemistry and Biology, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Dunn-Sims ER; Pfizer Worldwide Research and Development , Chemistry and Biology, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Hsu C; Pfizer Worldwide Research and Development , Chemistry and Biology, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Nawreen N; Pfizer Worldwide Research and Development , Chemistry and Biology, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Vanase-Frawley MA; Pfizer Worldwide Research and Development , Chemistry and Biology, Eastern Point Road, Groton, Connecticut 06340, United States.
  • O'Connor RE; Pfizer Worldwide Research and Development , Chemistry and Biology, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Schmidt CJ; Pfizer Worldwide Research and Development , Neuroscience Medicinal Chemistry and Neuroscience Research Unit, 610 Main Street, Cambridge, Massachusetts 02139, United States.
  • Dlugolenski K; Pfizer Worldwide Research and Development , Neuroscience Medicinal Chemistry and Neuroscience Research Unit, 610 Main Street, Cambridge, Massachusetts 02139, United States.
  • Stratman NC; Pfizer Worldwide Research and Development , Neuroscience Medicinal Chemistry and Neuroscience Research Unit, 610 Main Street, Cambridge, Massachusetts 02139, United States.
  • Majchrzak MJ; Pfizer Worldwide Research and Development , Chemistry and Biology, Eastern Point Road, Groton, Connecticut 06340, United States.
  • Kormos BL; Pfizer Worldwide Research and Development , Neuroscience Medicinal Chemistry and Neuroscience Research Unit, 610 Main Street, Cambridge, Massachusetts 02139, United States.
  • Nguyen DP; Pfizer Worldwide Research and Development , Pharmacokinetics, Dynamics, and Metabolism, 610 Main Street, Cambridge, Massachusetts 02139, United States.
  • Sawant-Basak A; Pfizer Worldwide Research and Development , Pharmacokinetics, Dynamics, and Metabolism, 610 Main Street, Cambridge, Massachusetts 02139, United States.
  • Mead AN; Pfizer Worldwide Research and Development , Chemistry and Biology, Eastern Point Road, Groton, Connecticut 06340, United States.
ACS Chem Neurosci ; 8(1): 165-177, 2017 01 18.
Article em En | MEDLINE | ID: mdl-27715007

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores de Dopamina D3 / Comportamento de Procura de Droga / Antagonistas dos Receptores de Dopamina D2 / Analgésicos Opioides Tipo de estudo: Prognostic_studies Limite: Animals / Humans / Male Idioma: En Revista: ACS Chem Neurosci Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores de Dopamina D3 / Comportamento de Procura de Droga / Antagonistas dos Receptores de Dopamina D2 / Analgésicos Opioides Tipo de estudo: Prognostic_studies Limite: Animals / Humans / Male Idioma: En Revista: ACS Chem Neurosci Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Estados Unidos