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Synthesis, biological evaluation, and molecular docking study of some new rohitukine analogs as protein tyrosine phosphatase 1B inhibitors.
Balaramnavar, V M; Srivastava, R; Varshney, S; Kumar, S; Rawat, A K; Chandasana, H; Chhonker, Y S; Bhatta, R S; Srivastava, A K; Gaikwad, A N; Lakshmi, V; Saxena, A K.
Afiliação
  • Balaramnavar VM; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Jankipuram, Extention Sector 10, Sitapur Road, Lucknow 226031, UP, India; Global Institute of Pharmaceutical Education and Research, Jaspur Road, Kashipur, Uttarakhand, India.
  • Srivastava R; Department of Biochemistry, CSIR-Central Drug Research Institute, Jankipuram Extention, Sector 10, Sitapur Road, Lucknow 226031, UP, India.
  • Varshney S; Department of Pharmacology, CSIR-Central Drug Research Institute, Jankipuram Extention Sector 10, Sitapur Road, Lucknow 226031, UP, India.
  • Kumar S; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Jankipuram, Extention Sector 10, Sitapur Road, Lucknow 226031, UP, India.
  • Rawat AK; Department of Biochemistry, CSIR-Central Drug Research Institute, Jankipuram Extention, Sector 10, Sitapur Road, Lucknow 226031, UP, India.
  • Chandasana H; Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Lucknow, India.
  • Chhonker YS; Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Lucknow, India.
  • Bhatta RS; Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Lucknow, India.
  • Srivastava AK; Department of Biochemistry, CSIR-Central Drug Research Institute, Jankipuram Extention, Sector 10, Sitapur Road, Lucknow 226031, UP, India.
  • Gaikwad AN; Department of Pharmacology, CSIR-Central Drug Research Institute, Jankipuram Extention Sector 10, Sitapur Road, Lucknow 226031, UP, India.
  • Lakshmi V; Department of Biochemistry, King George's Medical University, Lucknow 226003, UP, India.
  • Saxena AK; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Jankipuram, Extention Sector 10, Sitapur Road, Lucknow 226031, UP, India. Electronic address: anilsak@gmail.com.
Bioorg Chem ; 110: 104829, 2021 05.
Article em En | MEDLINE | ID: mdl-33773222

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piperidinas / Cromonas / Inibidores Enzimáticos / Proteína Tirosina Fosfatase não Receptora Tipo 1 Limite: Animals Idioma: En Revista: Bioorg Chem Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Índia País de publicação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piperidinas / Cromonas / Inibidores Enzimáticos / Proteína Tirosina Fosfatase não Receptora Tipo 1 Limite: Animals Idioma: En Revista: Bioorg Chem Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Índia País de publicação: Estados Unidos