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Novel topoisomerase II/EGFR dual inhibitors: design, synthesis and docking studies of naphtho[2',3':4,5]thiazolo[3,2-a]pyrimidine hybrids as potential anticancer agents with apoptosis inducing activity.
Mourad, Mai A E; Abo Elmaaty, Ayman; Zaki, Islam; Mourad, Ahmed A E; Hofni, Amal; Khodir, Ahmed E; Aboubakr, Esam M; Elkamhawy, Ahmed; Roh, Eun Joo; Al-Karmalawy, Ahmed A.
Afiliação
  • Mourad MAE; Medicinal Chemistry Department, Faculty of Pharmacy, Port-Said University, Port-Said, Egypt.
  • Abo Elmaaty A; Medicinal Chemistry Department, Faculty of Pharmacy, Port-Said University, Port-Said, Egypt.
  • Zaki I; Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Port-Said University, Port-Said, Egypt.
  • Mourad AAE; Pharmacology and Toxicology Department, Faculty of Pharmacy, Port-Said University, Port-Said, Egypt.
  • Hofni A; Department of Pharmacology and Toxicology, Faculty of Pharmacy, South Valley University, Qena, Egypt.
  • Khodir AE; Department of Pharmacology, Faculty of Pharmacy, Horus University, New Damietta, Egypt.
  • Aboubakr EM; Department of Pharmacology and Toxicology, Faculty of Pharmacy, South Valley University, Qena, Egypt.
  • Elkamhawy A; BK21 FOUR Team and Integrated Research Institute for Drug Development, College of Pharmacy, Dongguk University-Seoul, Goyang, Republic of Korea.
  • Roh EJ; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt.
  • Al-Karmalawy AA; Chemical and Biological Integrative Research Center, Korea Institute of Science and Technology (KIST), Seoul, Korea.
J Enzyme Inhib Med Chem ; 38(1): 2205043, 2023 Dec.
Article em En | MEDLINE | ID: mdl-37165800

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antineoplásicos Idioma: En Revista: J Enzyme Inhib Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Egito País de publicação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antineoplásicos Idioma: En Revista: J Enzyme Inhib Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Egito País de publicação: Reino Unido