Detalhe da pesquisa
1.
Sequential metabolism of AMG 487, a novel CXCR3 antagonist, results in formation of quinone reactive metabolites that covalently modify CYP3A4 Cys239 and cause time-dependent inhibition of the enzyme.
Drug Metab Dispos
; 40(7): 1429-40, 2012 Jul.
Artigo
em Inglês
| MEDLINE | ID: mdl-22517972