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1.

Direct Amidation of Esters by Ball Milling*.

Nicholson, William I; Barreteau, Fabien; Leitch, Jamie A; Payne, Riley; Priestley, Ian; Godineau, Edouard; Battilocchio, Claudio; Browne, Duncan L.

Angew Chem Int Ed Engl ; 60(40): 21868-21874, 2021 09 27.

Artigo em Inglês | MEDLINE | ID: mdl-34357668

2.

Direct Oxidation of Csp³ -H bonds using in Situ Generated Trifluoromethylated Dioxirane in Flow.

Lesieur, Mathieu; Battilocchio, Claudio; Labes, Ricardo; Jacq, Jérôme; Genicot, Christophe; Ley, Steven V; Pasau, Patrick.

Chemistry ; 25(5): 1203-1207, 2019 Jan 24.

Artigo em Inglês | MEDLINE | ID: mdl-30485562

3.

Building up a Continuous Flow Platform as an Enabler to the Preparation of Intermediates on Kilogram Scale.

Godineau, Edouard; Battilocchio, Claudio; Lal, Mukul.

Chimia (Aarau) ; 73(10): 828-831, 2019 Oct 30.

Artigo em Inglês | MEDLINE | ID: mdl-31645244

4.

Preparation of homoallylic amines via a three-component coupling process.

Ou, Xiaoxu; Labes, Ricardo; Battilocchio, Claudio; Ley, Steven V.

Org Biomol Chem ; 16(36): 6652-6654, 2018 09 19.

Artigo em Inglês | MEDLINE | ID: mdl-30183047

5.

Editorial.

Battilocchio, Claudio.

Chimia (Aarau) ; 77(5): 285, 2023 May 31.

Artigo em Inglês | MEDLINE | ID: mdl-38047822

6.

A Versatile Route to Unstable Diazo Compounds via Oxadiazolines and their Use in Aryl-Alkyl Cross-Coupling Reactions.

Greb, Andreas; Poh, Jian-Siang; Greed, Stephanie; Battilocchio, Claudio; Pasau, Patrick; Blakemore, David C; Ley, Steven V.

Angew Chem Int Ed Engl ; 56(52): 16602-16605, 2017 12 22.

Artigo em Inglês | MEDLINE | ID: mdl-29088512

7.

Rapid Asymmetric Synthesis of Disubstituted Allenes by Coupling of Flow-Generated Diazo Compounds and Propargylated Amines.

Poh, Jian-Siang; Makai, Szabolcs; von Keutz, Timo; Tran, Duc N; Battilocchio, Claudio; Pasau, Patrick; Ley, Steven V.

Angew Chem Int Ed Engl ; 56(7): 1864-1868, 2017 02 06.

Artigo em Inglês | MEDLINE | ID: mdl-28075518

8.

Visible Light Activation of Boronic Esters Enables Efficient Photoredox C(sp² )-C(sp³ ) Cross-Couplings in Flow.

Lima, Fabio; Kabeshov, Mikhail A; Tran, Duc N; Battilocchio, Claudio; Sedelmeier, Joerg; Sedelmeier, Gottfried; Schenkel, Berthold; Ley, Steven V.

Angew Chem Int Ed Engl ; 55(45): 14085-14089, 2016 11 02.

Artigo em Inglês | MEDLINE | ID: mdl-27709749

9.

The rapid synthesis of oxazolines and their heterogeneous oxidation to oxazoles under flow conditions.

Glöckner, Steffen; Tran, Duc N; Ingham, Richard J; Fenner, Sabine; Wilson, Zoe E; Battilocchio, Claudio; Ley, Steven V.

Org Biomol Chem ; 13(1): 207-14, 2015 Jan 07.

Artigo em Inglês | MEDLINE | ID: mdl-25370905

10.

Cyclopropanation using flow-generated diazo compounds.

Roda, Nuria M; Tran, Duc N; Battilocchio, Claudio; Labes, Ricardo; Ingham, Richard J; Hawkins, Joel M; Ley, Steven V.

Org Biomol Chem ; 13(9): 2550-4, 2015 Mar 07.

Artigo em Inglês | MEDLINE | ID: mdl-25600950

11.

A systems approach towards an intelligent and self-controlling platform for integrated continuous reaction sequences.

Ingham, Richard J; Battilocchio, Claudio; Fitzpatrick, Daniel E; Sliwinski, Eric; Hawkins, Joel M; Ley, Steven V.

Angew Chem Int Ed Engl ; 54(1): 144-8, 2015 Jan 02.

Artigo em Inglês | MEDLINE | ID: mdl-25377747

12.

Machine-Assisted Organic Synthesis.

Ley, Steven V; Fitzpatrick, Daniel E; Myers, Rebecca M; Battilocchio, Claudio; Ingham, Richard J.

Angew Chem Int Ed Engl ; 54(35): 10122-36, 2015 Aug 24.

Artigo em Inglês | MEDLINE | ID: mdl-26193360

13.

A Versatile Room-Temperature Route to Di- and Trisubstituted Allenes Using Flow-Generated Diazo Compounds.

Poh, Jian-Siang; Tran, Duc N; Battilocchio, Claudio; Hawkins, Joel M; Ley, Steven V.

Angew Chem Int Ed Engl ; 54(27): 7920-3, 2015 Jun 26.

Artigo em Inglês | MEDLINE | ID: mdl-26013774

14.

Enhancing the pharmacodynamic profile of a class of selective COX-2 inhibiting nitric oxide donors.

Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Consalvi, Sara; Di Capua, Angela; Calderone, Vincenzo; Martelli, Alma; Testai, Lara; Sautebin, Lidia; Rossi, Antonietta; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Giordani, Antonio; Persiani, Stefano; Colovic, Milena; Dovizio, Melania; Patrignani, Paola; Anzini, Maurizio.

Bioorg Med Chem ; 22(2): 772-86, 2014 Jan 15.

Artigo em Inglês | MEDLINE | ID: mdl-24373735

15.

Editorial.

Battilocchio, Claudio; Godineau, Edouard.

Chimia (Aarau) ; 73(10): 789, 2019 Oct 30.

Artigo em Inglês | MEDLINE | ID: mdl-31645238

16.

Integration of enabling methods for the automated flow preparation of piperazine-2-carboxamide.

Ingham, Richard J; Battilocchio, Claudio; Hawkins, Joel M; Ley, Steven V.

Beilstein J Org Chem ; 10: 641-52, 2014.

Artigo em Inglês | MEDLINE | ID: mdl-24778715

17.

A machine-assisted flow synthesis of SR48692: a probe for the investigation of neurotensin receptor-1.

Battilocchio, Claudio; Deadman, Benjamin J; Nikbin, Nikzad; Kitching, Matthew O; Baxendale, Ian R; Ley, Steven V.

Chemistry ; 19(24): 7917-30, 2013 Jun 10.

Artigo em Inglês | MEDLINE | ID: mdl-23592596

18.

A class of pyrrole derivatives endowed with analgesic/anti-inflammatory activity.

Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; Sautebin, Lidia; Pace, Simona; Rossi, Antonietta; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Schenone, Silvia; Giordani, Antonio; Di Francesco, Luigia; Patrignani, Paola; Biava, Mariangela.

Bioorg Med Chem ; 21(13): 3695-701, 2013 Jul 01.

Artigo em Inglês | MEDLINE | ID: mdl-23680444

19.

Correction to "Safety Considerations and Proposed Workflow for Laboratory Scale Chemical Synthesis by Ball Milling".

Priestley, Ian; Battilocchio, Claudio; Iosub, Andrei; Barreteau, Fabien; Bluck, Gavin W; Ling, Kenneth B; Ingram, Katharine; Ciaccia, Maria; Leitch, Jamie A; Browne, Duncan L.

Org Process Res Dev ; 27(6): 1154, 2023 Jun 16.

Artigo em Inglês | MEDLINE | ID: mdl-37342801

20.

MmpL3 is the cellular target of the antitubercular pyrrole derivative BM212.

La Rosa, Valentina; Poce, Giovanna; Canseco, Julio Ortiz; Buroni, Silvia; Pasca, Maria Rosalia; Biava, Mariangela; Raju, Ravikiran M; Porretta, Giulio Cesare; Alfonso, Salvatore; Battilocchio, Claudio; Javid, Babak; Sorrentino, Flavia; Ioerger, Thomas R; Sacchettini, James C; Manetti, Fabrizio; Botta, Maurizio; De Logu, Alessandro; Rubin, Eric J; De Rossi, Edda.

Antimicrob Agents Chemother ; 56(1): 324-31, 2012 Jan.

Artigo em Inglês | MEDLINE | ID: mdl-22024828

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Direct Amidation of Esters by Ball Milling*.

Direct Oxidation of Csp³ -H bonds using in Situ Generated Trifluoromethylated Dioxirane in Flow.

Building up a Continuous Flow Platform as an Enabler to the Preparation of Intermediates on Kilogram Scale.

Preparation of homoallylic amines via a three-component coupling process.

Editorial.

A Versatile Route to Unstable Diazo Compounds via Oxadiazolines and their Use in Aryl-Alkyl Cross-Coupling Reactions.

Rapid Asymmetric Synthesis of Disubstituted Allenes by Coupling of Flow-Generated Diazo Compounds and Propargylated Amines.

Visible Light Activation of Boronic Esters Enables Efficient Photoredox C(sp² )-C(sp³ ) Cross-Couplings in Flow.

The rapid synthesis of oxazolines and their heterogeneous oxidation to oxazoles under flow conditions.

Cyclopropanation using flow-generated diazo compounds.

A systems approach towards an intelligent and self-controlling platform for integrated continuous reaction sequences.

Machine-Assisted Organic Synthesis.

A Versatile Room-Temperature Route to Di- and Trisubstituted Allenes Using Flow-Generated Diazo Compounds.

Enhancing the pharmacodynamic profile of a class of selective COX-2 inhibiting nitric oxide donors.

Editorial.

Integration of enabling methods for the automated flow preparation of piperazine-2-carboxamide.

A machine-assisted flow synthesis of SR48692: a probe for the investigation of neurotensin receptor-1.

A class of pyrrole derivatives endowed with analgesic/anti-inflammatory activity.

Correction to "Safety Considerations and Proposed Workflow for Laboratory Scale Chemical Synthesis by Ball Milling".

MmpL3 is the cellular target of the antitubercular pyrrole derivative BM212.