Detalhe da pesquisa
1.
Tricyclic Diterpenoids Selectively Suppress Androgen Receptor-Positive Prostate Cancer Cells.
Molecules
; 28(12)2023 Jun 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-37375297
2.
5-Substituted 3, 3', 4', 7-tetramethoxyflavonoids - A novel class of potent DNA triplex specific binding ligands.
Bioorg Med Chem Lett
; 61: 128608, 2022 04 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-35143982
3.
Synthesis and biological evaluation of niclosamide PROTACs.
Bioorg Med Chem Lett
; 72: 128870, 2022 09 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-35772635
4.
An amide mimic of desTHPdactylolide: Total synthesis and antiproliferative evaluation.
Bioorg Med Chem Lett
; 40: 127970, 2021 05 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-33753258
5.
3-O-Carbamoyl-5,7,20-O-trimethylsilybins: Synthesis and Preliminary Antiproliferative Evaluation.
Molecules
; 26(21)2021 Oct 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-34770829
6.
Coinage metalides: a new class of excess electron compounds with high stability and large nonlinear optical responses.
Phys Chem Chem Phys
; 22(16): 8476-8484, 2020 Apr 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-32285081
7.
1-Chromonyl-5-Imidazolylpentadienone Demonstrates Anti-Cancer Action against TNBC and Exhibits Synergism with Paclitaxel.
Int J Mol Sci
; 21(16)2020 Aug 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-32806551
8.
New Zampanolide Mimics: Design, Synthesis, and Antiproliferative Evaluation.
Molecules
; 25(2)2020 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-31952332
9.
Second-Generation Androgen Receptor Antagonists as Hormonal Therapeutics for Three Forms of Prostate Cancer.
Molecules
; 25(10)2020 May 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-32456317
10.
Synthesis and antiproliferative evaluation of new zampanolide mimics.
Org Biomol Chem
; 17(15): 3830-3844, 2019 04 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-30924817
11.
Nitrogen-containing derivatives of O-tetramethylquercetin: Synthesis and biological profiles in prostate cancer cell models.
Bioorg Chem
; 87: 227-239, 2019 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-30904813
12.
Optimization of diarylpentadienones as chemotherapeutics for prostate cancer.
Bioorg Med Chem
; 26(16): 4751-4760, 2018 09 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-30121214
13.
Optimized synthesis and antiproliferative activity of desTHPdactylolides.
Bioorg Med Chem
; 26(12): 3514-3520, 2018 07 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-29784275
14.
Select ß- and γ-branched 1-alkylpyrazol-4-yl methylcarbamates exhibit high selectivity for inhibition of Anopheles gambiae versus human acetylcholinesterase.
Pestic Biochem Physiol
; 151: 32-39, 2018 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-30524149
15.
O-Aminoalkyl-O-Trimethyl-2,3-Dehydrosilybins: Synthesis and In Vitro Effects Towards Prostate Cancer Cells.
Molecules
; 23(12)2018 Nov 29.
Artigo
em Inglês
| MEDLINE | ID: mdl-30501133
16.
3-O-Substituted-3',4',5'-trimethoxyflavonols: Synthesis and cell-based evaluation as anti-prostate cancer agents.
Bioorg Med Chem
; 25(17): 4768-4777, 2017 09 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28760528
17.
5- or/and 20-O-alkyl-2,3-dehydrosilybins: Synthesis and biological profiles on prostate cancer cell models.
Bioorg Med Chem
; 25(17): 4845-4854, 2017 09 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28756013
18.
A new class of flavonol-based anti-prostate cancer agents: Design, synthesis, and evaluation in cell models.
Bioorg Med Chem Lett
; 26(17): 4241-5, 2016 09 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-27476422
19.
3-O-Alkyl-2,3-dehydrosilibinins: Two synthetic approaches and in vitro effects toward prostate cancer cells.
Bioorg Med Chem Lett
; 26(14): 3226-3231, 2016 07 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-27261177
20.
Design, synthesis, and biological evaluation of 1,9-diheteroarylnona-1,3,6,8-tetraen-5-ones as a new class of anti-prostate cancer agents.
Bioorg Med Chem
; 24(19): 4692-4700, 2016 10 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-27543391