Detalhe da pesquisa
1.
A Replicative In Vitro Assay for Drug Discovery against Leishmania donovani.
Antimicrob Agents Chemother
; 60(6): 3524-32, 2016 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-27021313
2.
Unravelling the rate of action of hits in the Leishmania donovani box using standard drugs amphotericin B and miltefosine.
PLoS Negl Trop Dis
; 11(5): e0005629, 2017 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-28542202
3.
The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold.
J Med Chem
; 60(16): 6880-6896, 2017 08 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-28806082
4.
Tetrahydro-2-naphthyl and 2-Indanyl Triazolopyrimidines Targeting Plasmodium falciparum Dihydroorotate Dehydrogenase Display Potent and Selective Antimalarial Activity.
J Med Chem
; 59(11): 5416-31, 2016 06 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-27127993
5.
Case Study of Small Molecules As Antimalarials: 2-Amino-1-phenylethanol (APE) Derivatives.
ACS Med Chem Lett
; 5(6): 657-61, 2014 Jun 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-24944739
6.
Correction to The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold.
J Med Chem
; 60(23): 9911, 2017 12 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-29164877
7.
Structure-guided lead optimization of triazolopyrimidine-ring substituents identifies potent Plasmodium falciparum dihydroorotate dehydrogenase inhibitors with clinical candidate potential.
J Med Chem
; 54(15): 5540-61, 2011 Aug 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-21696174
8.
Falcipain inhibitors: optimization studies of the 2-pyrimidinecarbonitrile lead series.
J Med Chem
; 53(16): 6129-52, 2010 Aug 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-20672841