Detalhe da pesquisa
1.
2,4-Diaminopyrimidine MK2 inhibitors. Part II: Structure-based inhibitor optimization.
Bioorg Med Chem Lett
; 20(1): 334-7, 2010 Jan 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-19926477
2.
3-amino-benzo[d]isoxazoles as novel multitargeted inhibitors of receptor tyrosine kinases.
J Med Chem
; 51(5): 1231-41, 2008 Mar 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-18260617
3.
Discovery of N-(4-(3-amino-1H-indazol-4-yl)phenyl)-N'-(2-fluoro-5-methylphenyl)urea (ABT-869), a 3-aminoindazole-based orally active multitargeted receptor tyrosine kinase inhibitor.
J Med Chem
; 50(7): 1584-97, 2007 Apr 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-17343372
4.
1,4-Dihydroindeno[1,2-c]pyrazoles with acetylenic side chains as novel and potent multitargeted receptor tyrosine kinase inhibitors with low affinity for the hERG ion channel.
J Med Chem
; 50(9): 2011-29, 2007 May 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-17425296
5.
Thienopyrimidine ureas as novel and potent multitargeted receptor tyrosine kinase inhibitors.
J Med Chem
; 48(19): 6066-83, 2005 Sep 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-16162008
6.
Synthesis and biological evaluation of 5-substituted 1,4-dihydroindeno[1,2-c]pyrazoles as multitargeted receptor tyrosine kinase inhibitors.
Bioorg Med Chem Lett
; 17(11): 3136-40, 2007 Jun 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-17391959
7.
Thienopyridine urea inhibitors of KDR kinase.
Bioorg Med Chem Lett
; 17(5): 1246-9, 2007 Mar 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-17188869
8.
Isothiazolopyrimidines and isoxazolopyrimidines as novel multi-targeted inhibitors of receptor tyrosine kinases.
Bioorg Med Chem Lett
; 16(16): 4326-30, 2006 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-16735117
9.
Hit-to-lead optimization of 1,4-dihydroindeno[1,2-c]pyrazoles as a novel class of KDR kinase inhibitors.
Bioorg Med Chem Lett
; 16(16): 4371-5, 2006 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-16750628
10.
1,4-Dihydroindeno[1,2-c]pyrazoles as novel multitargeted receptor tyrosine kinase inhibitors.
Bioorg Med Chem Lett
; 16(16): 4266-71, 2006 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-16759855
11.
Isoindolinone ureas: a novel class of KDR kinase inhibitors.
Bioorg Med Chem Lett
; 14(17): 4505-9, 2004 Sep 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-15357981