1.
Bioorg Med Chem Lett
; 12(10): 1405-11, 2002 May 20.
Artigo
em Inglês
| MEDLINE
| ID: mdl-11992787
RESUMO
The paper covers continuing efforts to discover novel, potent and selective oxytocin antagonists. Further benzofuran derivatives with potent oxytocin antagonist activity and good pharmacokinetic parameters are reported. Efforts to improve the in vivo activity of the series are described.