Detalhe da pesquisa
1.
Probing the Outstanding Local Hydrophobicity Increases in Peptide Sequences Induced by Incorporation of Trifluoromethylated Amino Acids.
Chembiochem
; 19(10): 1026-1030, 2018 05 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-29513394
2.
(R)-α-trifluoromethylalanine containing short peptide in the inhibition of amyloid peptide fibrillation.
Biopolymers
; 104(5): 601-10, 2015 Sep.
Artigo
em Inglês
| MEDLINE | ID: mdl-25968595
3.
An antedrug of the CXCL12 neutraligand blocks experimental allergic asthma without systemic effect in mice.
J Biol Chem
; 288(17): 11865-76, 2013 Apr 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-23449983
4.
A new pyrroline compound selective for I1-imidazoline receptors improves metabolic syndrome in rats.
J Pharmacol Exp Ther
; 346(3): 370-80, 2013 Sep.
Artigo
em Inglês
| MEDLINE | ID: mdl-23818682
5.
Methylation of imidazoline related compounds leads to loss of α2-adrenoceptor affinity. Synthesis and biological evaluation of selective I1 imidazoline receptor ligands.
Bioorg Med Chem
; 20(15): 4710-5, 2012 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-22750139
6.
From the Promiscuous Asenapine to Potent Fluorescent Ligands Acting at a Series of Aminergic G-Protein-Coupled Receptors.
J Med Chem
; 61(1): 174-188, 2018 01 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-29219316
7.
Discovery of a Locally and Orally Active CXCL12 Neutraligand (LIT-927) with Anti-inflammatory Effect in a Murine Model of Allergic Airway Hypereosinophilia.
J Med Chem
; 61(17): 7671-7686, 2018 09 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-30106292
8.
Synthesis and biological evaluation of 2-aryliminopyrrolidines as selective ligands for I1 imidazoline receptors: discovery of new sympatho-inhibitory hypotensive agents with potential beneficial effects in metabolic syndrome.
J Med Chem
; 58(2): 878-87, 2015 Jan 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-25521963
9.
Prodrugs of a CXC Chemokine-12 (CXCL12) Neutraligand Prevent Inflammatory Reactions in an Asthma Model in Vivo.
ACS Med Chem Lett
; 3(1): 10-4, 2012 Jan 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-24900366