Detalhe da pesquisa
1.
New 1H-1,2,4-Triazolyl Derivatives as Antimicrobial Agents.
Chem Biodivers
; 21(5): e202400316, 2024 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-38422224
2.
In silico Design, Synthesis and Biological Evaluation of Novel Thieno[3,2-d]pyrimidine Derivatives for Cancer Therapy - A Preliminary Study on the Inhibitory Potential towards ATR Kinase Domain and PIKK Family.
Chem Biodivers
; 21(3): e202302071, 2024 Mar.
Artigo
em Inglês
| MEDLINE | ID: mdl-38230843
3.
Design, Synthesis, and Evaluation of New Hybrid Derivatives of 5,6-Dihydro-4H-pyrrolo[3,2,1-ij]quinolin-2(1H)-one as Potential Dual Inhibitors of Blood Coagulation Factors Xa and XIa.
Molecules
; 29(2)2024 Jan 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-38257286
4.
Substituted furan sulfonamides as carbonic anhydrase inhibitors: Synthesis, biological and in silico studies.
Bioorg Chem
; 138: 106621, 2023 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-37257407
5.
Enzymes and Enzyme Inhibitors-Applications in Medicine and Diagnosis.
Int J Mol Sci
; 24(6)2023 Mar 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-36982319
6.
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors.
Int J Mol Sci
; 24(3)2023 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-36769114
7.
Antimicrobial Activity of Some Steroidal Hydrazones.
Molecules
; 28(3)2023 Jan 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-36770834
8.
Discovery of Novel EGFR Inhibitor Targeting Wild-Type and Mutant Forms of EGFR: In Silico and In Vitro Study.
Molecules
; 28(7)2023 Mar 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-37049777
9.
New Bicyclic Pyridine-Based Hybrids Linked to the 1,2,3-Triazole Unit: Synthesis via Click Reaction and Evaluation of Neurotropic Activity and Molecular Docking.
Molecules
; 28(3)2023 Jan 17.
Artigo
em Inglês
| MEDLINE | ID: mdl-36770592
10.
Identification of Novel Cyclooxygenase-1 Selective Inhibitors of Thiadiazole-Based Scaffold as Potent Anti-Inflammatory Agents with Safety Gastric and Cytotoxic Profile.
Molecules
; 28(8)2023 Apr 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-37110650
11.
New Hybrid Tetrahydropyrrolo[3,2,1-ij]quinolin-1-ylidene-2-thioxothiazolidin-4-ones as New Inhibitors of Factor Xa and Factor XIa: Design, Synthesis, and In Silico and Experimental Evaluation.
Molecules
; 28(9)2023 May 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-37175261
12.
Developing New Treatments for COVID-19 through Dual-Action Antiviral/Anti-Inflammatory Small Molecules and Physiologically Based Pharmacokinetic Modeling.
Int J Mol Sci
; 23(14)2022 07 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-35887353
13.
Synthesis of 1-Amino-3-oxo-2,7-naphthyridines via Smiles Rearrangement: A New Approach in the Field of Chemistry of Heterocyclic Compounds.
Int J Mol Sci
; 23(11)2022 May 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-35682584
14.
Benzothiazole and Chromone Derivatives as Potential ATR Kinase Inhibitors and Anticancer Agents.
Molecules
; 27(14)2022 Jul 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-35889508
15.
Thiazolidin-4-Ones as Potential Antimicrobial Agents: Experimental and In Silico Evaluation.
Molecules
; 27(6)2022 Mar 16.
Artigo
em Inglês
| MEDLINE | ID: mdl-35335296
16.
Thiazole/Thiadiazole/Benzothiazole Based Thiazolidin-4-One Derivatives as Potential Inhibitors of Main Protease of SARS-CoV-2.
Molecules
; 27(7)2022 Mar 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-35408577
17.
Discovery of 5-Methylthiazole-Thiazolidinone Conjugates as Potential Anti-Inflammatory Agents: Molecular Target Identification and In Silico Studies.
Molecules
; 27(23)2022 Nov 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-36500230
18.
A Multifield Study on Dimethyl Acetylenedicarboxylate: A Reagent Able to Build a New Cycle on Diaminoimidazoles.
Molecules
; 27(10)2022 May 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-35630803
19.
Synthesis, Biological Evaluation and Molecular Docking Studies of 5-Indolylmethylen-4-oxo-2-thioxothiazolidine Derivatives.
Molecules
; 27(3)2022 Feb 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-35164333
20.
2-Aryl-3-(6-trifluoromethoxy)benzo[d]thiazole-based thiazolidinone hybrids as potential anti-infective agents: Synthesis, biological evaluation and molecular docking studies.
Bioorg Med Chem Lett
; 32: 127718, 2021 01 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-33253880