Detalhe da pesquisa
1.
A Stereocontrolled Synthesis of a Phosphorothioate Cyclic Dinucleotide-Based STING Agonist.
J Org Chem
; 86(13): 8851-8861, 2021 07 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-34126006
2.
Substituted diaryl ether compounds as retinoic acid-related orphan Receptor-γt (RORγt) agonists.
Bioorg Med Chem Lett
; 35: 127778, 2021 03 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-33422603
3.
Substituted benzyloxytricyclic compounds as retinoic acid-related orphan receptor gamma t (RORγt) agonists.
Bioorg Med Chem Lett
; 30(12): 127204, 2020 06 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-32334911
4.
Heterobicyclic inhibitors of transforming growth factor beta receptor I (TGFßRI).
Bioorg Med Chem
; 26(5): 1026-1034, 2018 03 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-29422332
5.
Diphenylpyridylethanamine (DPPE)-based aminoheterocycles as cholesteryl ester transfer protein inhibitors.
Bioorg Med Chem Lett
; 24(3): 860-4, 2014 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-24424134
6.
Identification and optimization of small molecule antagonists of vasoactive intestinal peptide receptor-1 (VIPR1).
Bioorg Med Chem Lett
; 22(6): 2287-90, 2012 Mar 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22365758
7.
Pyrrolo[1,2-f]triazines as JAK2 inhibitors: achieving potency and selectivity for JAK2 over JAK3.
Bioorg Med Chem Lett
; 21(5): 1425-8, 2011 Mar 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21282055
8.
Design and synthesis of a G-protein-coupled receptor antagonist library of aryloxyalkanolamines using a polymer-supported acyclic acetal linker.
J Comb Chem
; 11(1): 72-82, 2009.
Artigo
em Inglês
| MEDLINE | ID: mdl-19086798
9.
Discovery of a Lead Triphenylethanamine Cholesterol Ester Transfer Protein (CETP) Inhibitor.
ACS Med Chem Lett
; 10(6): 911-916, 2019 Jun 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-31223447
10.
2-Arylbenzoxazoles as novel cholesteryl ester transfer protein inhibitors: optimization via array synthesis.
Bioorg Med Chem Lett
; 18(8): 2640-4, 2008 Apr 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-18374566
11.
Triphenylethanamine Derivatives as Cholesteryl Ester Transfer Protein Inhibitors: Discovery of N-[(1R)-1-(3-Cyclopropoxy-4-fluorophenyl)-1-[3-fluoro-5-(1,1,2,2-tetrafluoroethoxy)phenyl]-2-phenylethyl]-4-fluoro-3-(trifluoromethyl)benzamide (BMS-795311).
J Med Chem
; 58(22): 9010-26, 2015 Nov 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-26524347
12.
Preparation of 2,7-diaminosubstituted-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonitriles by solid-phase synthesis.
J Comb Chem
; 10(1): 28-30, 2008.
Artigo
em Inglês
| MEDLINE | ID: mdl-17994705
13.
Diphenylpyridylethanamine (DPPE) derivatives as cholesteryl ester transfer protein (CETP) inhibitors.
J Med Chem
; 55(13): 6162-75, 2012 Jul 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-22650305