Detalhe da pesquisa
1.
Discovery and optimization of novel constrained pyrrolopyridone BET family inhibitors.
Bioorg Med Chem Lett
; 28(10): 1804-1810, 2018 06 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-29678460
2.
Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors.
J Med Chem
; 60(9): 3828-3850, 2017 05 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-28368119
3.
Phenoxyphenyl sulfone N-formylhydroxylamines (retrohydroxamates) as potent, selective, orally bioavailable matrix metalloproteinase inhibitors.
J Med Chem
; 45(1): 219-32, 2002 Jan 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-11754593
4.
Expression and functional characterization of recombinant human HDAC1 and HDAC3.
Life Sci
; 74(22): 2693-705, 2004 Apr 16.
Artigo
em Inglês
| MEDLINE | ID: mdl-15043985
5.
Alpha-keto amides as inhibitors of histone deacetylase.
Bioorg Med Chem Lett
; 13(19): 3331-5, 2003 Oct 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-12951120