Detalhe da pesquisa
1.
Discovery of novel, non-acidic mPGES-1 inhibitors by virtual screening with a multistep protocol.
Bioorg Med Chem
; 23(15): 4839-4845, 2015 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-26088337
2.
Honokiol: a non-adipogenic PPARγ agonist from nature.
Biochim Biophys Acta
; 1830(10): 4813-9, 2013 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-23811337
3.
Tetra- and pentacyclic triterpene acids from the ancient anti-inflammatory remedy frankincense as inhibitors of microsomal prostaglandin E(2) synthase-1.
J Nat Prod
; 77(6): 1445-51, 2014 Jun 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-24844534
4.
Polyyne hybrid compounds from Notopterygium incisum with peroxisome proliferator-activated receptor gamma agonistic effects.
J Nat Prod
; 77(11): 2513-21, 2014 Nov 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-25333853
5.
Identification of isosilybin a from milk thistle seeds as an agonist of peroxisome proliferator-activated receptor gamma.
J Nat Prod
; 77(4): 842-7, 2014 Apr 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-24597776
6.
Pharmacophore-based discovery of a novel cytosolic phospholipase A(2)α inhibitor.
Bioorg Med Chem Lett
; 22(2): 1202-7, 2012 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22192589
7.
Discovery of a novel IKK-ß inhibitor by ligand-based virtual screening techniques.
Bioorg Med Chem Lett
; 21(1): 577-83, 2011 Jan 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21078555
8.
Pharmacophore-based discovery of FXR agonists. Part I: Model development and experimental validation.
Bioorg Med Chem
; 19(23): 7168-80, 2011 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-22018919
9.
Discovery of carbazole derivatives as novel allosteric MEK inhibitors by pharmacophore modeling and virtual screening.
Eur J Med Chem
; 178: 802-817, 2019 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-31252285
10.
Molecular Docking, Molecular Dynamics, and Structure-Activity Relationship Explorations of 14-Oxygenated N-Methylmorphinan-6-ones as Potent µ-Opioid Receptor Agonists.
ACS Chem Neurosci
; 8(6): 1327-1337, 2017 06 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-28125215
11.
Synthesis, Pharmacology, and Molecular Docking Studies on 6-Desoxo-N-methylmorphinans as Potent µ-Opioid Receptor Agonists.
J Med Chem
; 60(22): 9407-9412, 2017 11 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-29053268
12.
Potent inhibition of human 5-lipoxygenase and microsomal prostaglandin E2 synthase-1 by the anti-carcinogenic and anti-inflammatory agent embelin.
Biochem Pharmacol
; 86(4): 476-86, 2013 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-23623753
13.
Polyacetylenes from Notopterygium incisum--new selective partial agonists of peroxisome proliferator-activated receptor-gamma.
PLoS One
; 8(4): e61755, 2013.
Artigo
em Inglês
| MEDLINE | ID: mdl-23630612
14.
Discovery of depsides and depsidones from lichen as potent inhibitors of microsomal prostaglandin E2 synthase-1 using pharmacophore models.
ChemMedChem
; 7(12): 2077-81, 2012 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-23109349
15.
Pharmacophore modeling and virtual screening for novel acidic inhibitors of microsomal prostaglandin E2 synthase-1 (mPGES-1).
J Med Chem
; 54(9): 3163-74, 2011 May 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-21466167