1.
Bioorg Med Chem Lett
; 18(16): 4731-5, 2008 Aug 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-18640834
RESUMO
A new method for solid phase parallel synthesis of chemically and conformationally diverse macrocyclic peptidomimetics is reported. A key feature of the method is access to broad chemical and conformational diversity. Synthesis and mechanistic studies on the macrocyclization step are reported.