Pesquisa | Biblioteca Virtual em Saúde

1.

Multiplexed cellular profiling identifies an organoselenium compound as an inhibitor of CRM1-mediated nuclear export.

Jimenez, Lucia; Mayoral-Varo, Victor; Amenábar, Carlos; Ortega, Judit; Sequeira, João G N; Machuqueiro, Miguel; Mourato, Cristiana; Silvestri, Romano; Angeli, Andrea; Carta, Fabrizio; Supuran, Claudiu T; Megías, Diego; Ferreira, Bibiana I; Link, Wolfgang.

Traffic ; 23(12): 587-599, 2022 12.

Artigo em Inglês | MEDLINE | ID: mdl-36353954

2.

Boron-containing carbonic anhydrases inhibitors.

Giovannuzzi, Simone; Nikitjuka, Anna; Pereira Resende, Bruna Rafaela; Smietana, Michael; Nocentini, Alessio; Supuran, Claudiu T; Winum, Jean-Yves.

Bioorg Chem ; 143: 106976, 2024 Feb.

Artigo em Inglês | MEDLINE | ID: mdl-38000350

3.

A comparative study of diaryl urea molecules with and without sulfonamide group on Carbonic anhydrase IX and XII inhibition and its consequence on breast cancer cells.

Debnath, Joy; Keshamasetthy, Dhananjaya; Combs, Jacob; Leon, Katherine; Vullo, Daniela; Chatterjee, Abhijit; McKenna, Robert; Supuran, Claudiu T.

Bioorg Chem ; 145: 107192, 2024 Apr.

Artigo em Inglês | MEDLINE | ID: mdl-38382393

4.

Novel 2-(hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide based thiosemicarbazides as potent and selective inhibitors of tumor-associated human carbonic anhydrase IX and XII: Synthesis, cytotoxicity, and molecular modelling studies.

Demir-Yazici, Kübra; Trawally, Muhammed; Bua, Silvia; Öztürk-Civelek, Dilek; Akdemir, Atilla; Supuran, Claudiu T; Güzel-Akdemir, Özlen.

Bioorg Chem ; 144: 107096, 2024 Mar.

Artigo em Inglês | MEDLINE | ID: mdl-38290186

5.

Identification of thienopyrimidine derivatives tethered with sulfonamide and other moieties as carbonic anhydrase inhibitors: Design, synthesis and anti-proliferative activity.

Higazy, Samah; Samir, Nermin; El-Khouly, Ahmed; Giovannuzzi, Simone; Begines, Paloma; Gaber, Hatem M; Supuran, Claudiu T; Abouzid, Khaled A M.

Bioorg Chem ; 144: 107089, 2024 Mar.

Artigo em Inglês | MEDLINE | ID: mdl-38237393

6.

Coumarins-lipophilic cations conjugates: Efficient mitocans targeting carbonic anhydrases.

Fuentes-Aguilar, Alma; González-Bakker, Aday; Jovanovic, Mirna; Stojanov, Sofija Jovanovic; Puerta, Adrián; Gargano, Adriana; Dinic, Jelena; Vega-Báez, José L; Merino-Montiel, Penélope; Montiel-Smith, Sara; Alcaro, Stefano; Nocentini, Alessio; Pesic, Milica; Supuran, Claudiu T; Padrón, José M; Fernández-Bolaños, José G; López, Óscar.

Bioorg Chem ; 145: 107168, 2024 Apr.

Artigo em Inglês | MEDLINE | ID: mdl-38354500

7.

Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids.

Abdoli, Morteza; Bonardi, Alessandro; Gratteri, Paola; Supuran, Claudiu T; Zalubovskis, Raivis.

J Enzyme Inhib Med Chem ; 39(1): 2335927, 2024 Dec.

Artigo em Inglês | MEDLINE | ID: mdl-38606915

8.

In-vitro and in-silico investigations of SLC-0111 hydrazinyl analogs as human carbonic anhydrase I, II, IX, and XII inhibitors.

Sharma, Vikas; Vats, Lalit; Giovannuzzi, Simone; Mohan, Brij; Supuran, Claudiu T; Sharma, Pawan K.

Arch Pharm (Weinheim) ; : e2400157, 2024 May 07.

Artigo em Inglês | MEDLINE | ID: mdl-38713910

9.

Chemistry of heterocycles as carbonic anhydrase inhibitors: A pathway to novel research in medicinal chemistry review.

Bendi, Anjaneyulu; Kataria, Sweety; Singh, Lakhwinder; Kennedy, John F; Supuran, Claudiu T; Raghav, Neera.

Arch Pharm (Weinheim) ; : e2400073, 2024 Apr 29.

Artigo em Inglês | MEDLINE | ID: mdl-38683875

10.

Sulfonamide-incorporated bis(α-aminophosphonates) as promising carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and X-ray crystallographic studies.

Sobati, Marjan; Abdoli, Morteza; Angeli, Andrea; Bonardi, Alessandro; Ferraroni, Marta; Supuran, Claudiu T; Zalubovskis, Raivis.

Arch Pharm (Weinheim) ; : e2400038, 2024 Mar 18.

Artigo em Inglês | MEDLINE | ID: mdl-38498884

11.

1,2,3-Triazole-based esters and carboxylic acids as nonclassical carbonic anhydrase inhibitors capable of cathepsin B inhibition.

Siwach, Kiran; Rani, Manishita; Vats, Lalit; Giovannuzzi, Simone; Paul, Avijit Kumar; Brahma, Mettle; Kumari, Neetu; Maruthi, Mulaka; Raghav, Neera; Supuran, Claudiu T; Sharma, Pawan K.

Arch Pharm (Weinheim) ; 357(3): e2300372, 2024 Mar.

Artigo em Inglês | MEDLINE | ID: mdl-38012535

12.

Design, synthesis, and biological evaluation of 3-benzenesulfonamide-linked 3-hydrazinoisatin derivatives as carbonic anhydrase inhibitors.

Swain, Baijayantimala; Marde, Vaibhav S; Singh, Priti; Angeli, Andrea; Khan, Abrar; Yaddanapudi, Venkata M; Ullah, Qasim; Supuran, Claudiu T; Arifuddin, Mohammed.

Arch Pharm (Weinheim) ; : e2300718, 2024 Mar 11.

Artigo em Inglês | MEDLINE | ID: mdl-38466120

13.

Exploring rhodanine linked enamine-carbohydrazide derivatives as mycobacterial carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and molecular docking studies.

Maddipatla, Sarvan; Bakchi, Bulti; Gadhave, Rutuja Rama; Ammara, Andrea; Sau, Shashikanta; Rani, Bandela; Nanduri, Srinivas; Kalia, Nitin Pal; Supuran, Claudiu T; Yaddanapudi, Venkata Madhavi.

Arch Pharm (Weinheim) ; : e2400064, 2024 Mar 18.

Artigo em Inglês | MEDLINE | ID: mdl-38498883

14.

Identification of 3-(5-cyano-6-oxo-pyridin-2-yl)benzenesulfonamides as novel anticancer agents endowed with EGFR inhibitory activity.

Shaldam, Moataz A; Khalil, Ahmed F; Almahli, Hadia; Jaballah, Maiy Y; Angeli, Andrea; Khaleel, Eman F; Badi, Rehab Mustafa; Elkaeed, Eslam B; Supuran, Claudiu T; Eldehna, Wagdy M; Tawfik, Haytham O.

Arch Pharm (Weinheim) ; 357(1): e2300449, 2024 Jan.

Artigo em Inglês | MEDLINE | ID: mdl-37828544

15.

Novel sulfonamide-phosphonate conjugates as carbonic anhydrase isozymes inhibitors.

Bekheit, Mohamed S; Sabry, Eman; Mohamed, Hanan A; Ewies, Ewies F; Kariuki, Benson M; Fouad, Marwa A; Vullo, Daniela; Supuran, Claudiu T.

Drug Dev Res ; 85(1): e22135, 2024 Feb.

Artigo em Inglês | MEDLINE | ID: mdl-37997034

16.

Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains.

Bua, Silvia; Bonardi, Alessandro; Mük, Georgiana Ramona; Nocentini, Alessio; Gratteri, Paola; Supuran, Claudiu T.

Int J Mol Sci ; 25(5)2024 Feb 23.

Artigo em Inglês | MEDLINE | ID: mdl-38473830

17.

Leveraging SARS-CoV-2 Main Protease (M^pro) for COVID-19 Mitigation with Selenium-Based Inhibitors.

De Luca, Viviana; Angeli, Andrea; Nocentini, Alessio; Gratteri, Paola; Pratesi, Silvia; Tanini, Damiano; Carginale, Vincenzo; Capperucci, Antonella; Supuran, Claudiu T; Capasso, Clemente.

Int J Mol Sci ; 25(2)2024 Jan 12.

Artigo em Inglês | MEDLINE | ID: mdl-38256046

18.

Mitochondrial carbonic anhydrase VA and VB: properties and roles in health and disease.

Aspatwar, Ashok; Supuran, Claudiu T; Waheed, Abdul; Sly, William S; Parkkila, Seppo.

J Physiol ; 601(2): 257-274, 2023 01.

Artigo em Inglês | MEDLINE | ID: mdl-36464834

19.

A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation.

Supuran, Claudiu T.

Bioorg Med Chem Lett ; 93: 129411, 2023 09 01.

Artigo em Inglês | MEDLINE | ID: mdl-37507055

20.

Potent and selective carbonic anhydrase inhibition activities of pyrazolones bearing benzenesulfonamides.

Akocak, Suleyman; Lolak, Nebih; Giovannuzzi, Simone; Supuran, Claudiu T.

Bioorg Med Chem Lett ; 95: 129479, 2023 10 15.

Artigo em Inglês | MEDLINE | ID: mdl-37704010

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