Detalhe da pesquisa
1.
Identification of 2-((2,3-dihydrobenzo[b][1,4]dioxin-6-yl)amino)-N-phenylpropanamides as a novel class of potent DprE1 inhibitors.
Bioorg Med Chem Lett
; 30(12): 127192, 2020 06 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-32312582
2.
Covalent hits and where to find them.
SLAS Discov
; 29(3): 100142, 2024 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-38278484
3.
Design and Evaluation of a Low Hydrogen Bond Donor Count Fragment Screening Set to Aid Hit Generation of PROTACs Intended for Oral Delivery.
J Med Chem
; 66(11): 7594-7604, 2023 06 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-37224440
4.
Put a ring on it: application of small aliphatic rings in medicinal chemistry.
RSC Med Chem
; 12(4): 448-471, 2021 Apr 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-33937776
5.
Mycobacterium tuberculosis Decaprenylphosphoryl-ß-d-ribose Oxidase Inhibitors: Expeditious Reconstruction of Suboptimal Hits into a Series with Potent in Vivo Activity.
J Med Chem
; 63(5): 2557-2576, 2020 03 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-31922409
6.
Chemoselective Sequential Click Ligations Directed by Enhanced Reactivity of an Aromatic Ynamine.
Org Lett
; 18(7): 1694-7, 2016 Apr 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-27001375
7.
Chemoselective Sequential Click Ligations Directed by Enhanced Reactivity of an Aromatic Ynamine.
Org Lett
; 18(9): 2326, 2016 05 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-27090999