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Full antagonism of the estrogen receptor without a prototypical ligand side chain.
Srinivasan, Sathish; Nwachukwu, Jerome C; Bruno, Nelson E; Dharmarajan, Venkatasubramanian; Goswami, Devrishi; Kastrati, Irida; Novick, Scott; Nowak, Jason; Cavett, Valerie; Zhou, Hai-Bing; Boonmuen, Nittaya; Zhao, Yuechao; Min, Jian; Frasor, Jonna; Katzenellenbogen, Benita S; Griffin, Patrick R; Katzenellenbogen, John A; Nettles, Kendall W.
Afiliação
  • Srinivasan S; Department of Cancer Biology, The Scripps Research Institute, Jupiter, Florida, USA.
  • Nwachukwu JC; Department of Cancer Biology, The Scripps Research Institute, Jupiter, Florida, USA.
  • Bruno NE; Department of Cancer Biology, The Scripps Research Institute, Jupiter, Florida, USA.
  • Dharmarajan V; Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida, USA.
  • Goswami D; Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida, USA.
  • Kastrati I; Department of Physiology and Biophysics, University of Illinois, Chicago, Illinois, USA.
  • Novick S; Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida, USA.
  • Nowak J; Department of Cancer Biology, The Scripps Research Institute, Jupiter, Florida, USA.
  • Cavett V; Department of Cancer Biology, The Scripps Research Institute, Jupiter, Florida, USA.
  • Zhou HB; Key Laboratory of Combinatorial Biosynthesis and Drug Discovery (Wuhan University), Ministry of Education, State Key Laboratory of Virology, Wuhan University School of Pharmaceutical Sciences, Wuhan, China.
  • Boonmuen N; Department of Molecular and Integrative Physiology, University of Illinois, Urbana, Illinois, USA.
  • Zhao Y; Department of Molecular and Integrative Physiology, University of Illinois, Urbana, Illinois, USA.
  • Min J; Department of Chemistry, University of Illinois, Urbana, Illinois, USA.
  • Frasor J; Department of Physiology and Biophysics, University of Illinois, Chicago, Illinois, USA.
  • Katzenellenbogen BS; Department of Molecular and Integrative Physiology, University of Illinois, Urbana, Illinois, USA.
  • Griffin PR; Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida, USA.
  • Katzenellenbogen JA; Department of Chemistry, University of Illinois, Urbana, Illinois, USA.
  • Nettles KW; Department of Cancer Biology, The Scripps Research Institute, Jupiter, Florida, USA.
Nat Chem Biol ; 13(1): 111-118, 2017 01.
Article em En | MEDLINE | ID: mdl-27870835

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Limite: Female / Humans Idioma: En Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Limite: Female / Humans Idioma: En Ano de publicação: 2017 Tipo de documento: Article