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Characterization of new, efficient Mycobacterium tuberculosis topoisomerase-I inhibitors and their interaction with human ABC multidrug transporters.
Temesszentandrási-Ambrus, Csilla; Tóth, Szilárd; Verma, Rinkee; Bánhegyi, Péter; Szabadkai, István; Baska, Ferenc; Szántai-Kis, Csaba; Hartkoorn, Ruben C; Lingerfelt, Mary A; Sarkadi, Balázs; Szakács, Gergely; Orfi, László; Nagaraja, Valakunja; Ekins, Sean; Telbisz, Ágnes.
Afiliação
  • Temesszentandrási-Ambrus C; Institute of Enzymology, RCNS-HAS, Budapest, Hungary.
  • Tóth S; Molecular Medicine Doctoral School, Semmelweis University, Budapest, Hungary.
  • Verma R; Institute of Enzymology, RCNS-HAS, Budapest, Hungary.
  • Bánhegyi P; Department of Microbiology and Cell Biology, Indian Institute of Science, Bangalore, India.
  • Szabadkai I; Vichem Chemie Research Ltd., Budapest, Hungary.
  • Baska F; Vichem Chemie Research Ltd., Budapest, Hungary.
  • Szántai-Kis C; Vichem Chemie Research Ltd., Budapest, Hungary.
  • Hartkoorn RC; Vichem Chemie Research Ltd., Budapest, Hungary.
  • Lingerfelt MA; Chemical Biology of Antibiotics, Center for Infection and Immunity, Inserm, CNRS, Institut Pasteur de Lille, Université de Lille, Lille, France.
  • Sarkadi B; Collaborations Pharmaceuticals, Inc., Raleigh, United States of America.
  • Szakács G; Institute of Enzymology, RCNS-HAS, Budapest, Hungary.
  • Orfi L; Institute of Enzymology, RCNS-HAS, Budapest, Hungary.
  • Nagaraja V; Vichem Chemie Research Ltd., Budapest, Hungary.
  • Ekins S; Department of Pharmaceutical Chemistry, Semmelweis University, Budapest, Hungary.
  • Telbisz Á; Department of Microbiology and Cell Biology, Indian Institute of Science, Bangalore, India.
PLoS One ; 13(9): e0202749, 2018.
Article em En | MEDLINE | ID: mdl-30183750

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Limite: Animals / Humans Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Limite: Animals / Humans Idioma: En Ano de publicação: 2018 Tipo de documento: Article