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Lerisetron Analogues with Antimalarial Properties: Synthesis, Structure-Activity Relationship Studies, and Biological Assessment.
Mueller, Rudolf; Reddy, Virsinha; Nchinda, Aloysius T; Mebrahtu, Fanuel; Taylor, Dale; Lawrence, Nina; Tanner, Lloyd; Barnabe, Marine; Eyermann, Charles J; Zou, Bin; Kondreddi, Ravinder R; Lakshminarayana, Suresh B; Rottmann, Matthias; Street, Leslie J; Chibale, Kelly.
Afiliação
  • Mueller R; Drug Discovery and Development Centre (H3D), Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa.
  • Reddy V; Drug Discovery and Development Centre (H3D), Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa.
  • Nchinda AT; Drug Discovery and Development Centre (H3D), Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa.
  • Mebrahtu F; Drug Discovery and Development Centre (H3D), Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa.
  • Taylor D; Drug Discovery and Development Centre (H3D), Division of Clinical Pharmacology, Department of Medicine, University of Cape Town, Observatory 7925, South Africa.
  • Lawrence N; Drug Discovery and Development Centre (H3D), Division of Clinical Pharmacology, Department of Medicine, University of Cape Town, Observatory 7925, South Africa.
  • Tanner L; Drug Discovery and Development Centre (H3D), Division of Clinical Pharmacology, Department of Medicine, University of Cape Town, Observatory 7925, South Africa.
  • Barnabe M; Drug Discovery and Development Centre (H3D), Division of Clinical Pharmacology, Department of Medicine, University of Cape Town, Observatory 7925, South Africa.
  • Eyermann CJ; Drug Discovery and Development Centre (H3D), Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa.
  • Zou B; Shanghai Blueray Biopharma Co. LTD, Block 3, 576 Libing Road, Pudong New District, Shanghai 201301, China.
  • Kondreddi RR; PJS Pharma Pvt. Ltd., Plot No. 103/1, Phase II, IDA Cherlapally, Hyderabad 500051, India.
  • Lakshminarayana SB; Novartis Institute for Tropical Diseases, 5300 Chiron Way, Emeryville, California 94608, United States.
  • Rottmann M; Department of Medical Parasitology and Infection Biology, Swiss Tropical and Public Health Institute, CH-4051 Basel, Switzerland.
  • Street LJ; University of Basel, 4002 Basel, Switzerland.
  • Chibale K; Drug Discovery and Development Centre (H3D), Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa.
ACS Omega ; 5(12): 6967-6982, 2020 Mar 31.
Article em En | MEDLINE | ID: mdl-32258933

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article