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Discovery of Potent and Selective 7-Azaindole Isoindolinone-Based PI3Kγ Inhibitors.
Miles, Dillon H; Yan, Xuelei; Thomas-Tran, Rhiannon; Fournier, Jeremy; Sharif, Ehesan U; Drew, Samuel L; Mata, Guillaume; Lawson, Kenneth V; Ginn, Elaine; Wong, Kent; Soni, Divyank; Dhanota, Puja; Shaqfeh, Stefan G; Meleza, Cesar; Chen, Ada; Pham, Amber T; Park, Timothy; Swinarski, Debbie; Banuelos, Jesus; Schindler, Ulrike; Walters, Matthew J; Walker, Nigel P; Zhao, Xiaoning; Young, Stephen W; Chen, Jie; Jin, Lixia; Leleti, Manmohan Reddy; Powers, Jay P; Jeffrey, Jenna L.
Afiliação
  • Miles DH; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Yan X; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Thomas-Tran R; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Fournier J; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Sharif EU; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Drew SL; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Mata G; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Lawson KV; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Ginn E; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Wong K; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Soni D; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Dhanota P; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Shaqfeh SG; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Meleza C; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Chen A; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Pham AT; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Park T; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Swinarski D; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Banuelos J; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Schindler U; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Walters MJ; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Walker NP; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Zhao X; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Young SW; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Chen J; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Jin L; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Leleti MR; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Powers JP; Arcus Biosciences, Inc., Hayward, California 94545, United States.
  • Jeffrey JL; Arcus Biosciences, Inc., Hayward, California 94545, United States.
ACS Med Chem Lett ; 11(11): 2244-2252, 2020 Nov 12.
Article em En | MEDLINE | ID: mdl-33214836

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article