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Translatability of in vitro Inhibition Potency to in vivo P-Glycoprotein Mediated Drug Interaction Risk.
Lazzaro, Sarah; West, Mark A; Eatemadpour, Soraya; Feng, Bo; Varma, Manthena V S; Rodrigues, A David; Temesszentandrási-Ambrus, Csilla; Kovács-Hajdu, Péter; Nerada, Zsuzsanna; Gáborik, Zsuzsanna; Costales, Chester.
Afiliação
  • Lazzaro S; Medicine Design-PDM, Worldwide Research and Development, Pfizer Inc., Groton, Connecticut, USA.
  • West MA; Medicine Design-PDM, Worldwide Research and Development, Pfizer Inc., Groton, Connecticut, USA.
  • Eatemadpour S; Medicine Design-PDM, Worldwide Research and Development, Pfizer Inc., Groton, Connecticut, USA; Eurofins, Research Triangle Park, North Carolina, USA.
  • Feng B; Medicine Design-PDM, Worldwide Research and Development, Pfizer Inc., Groton, Connecticut, USA; DMPK, Vertex Pharmaceuticals, Boston, Massachusetts, USA.
  • Varma MVS; Medicine Design-PDM, Worldwide Research and Development, Pfizer Inc., Groton, Connecticut, USA.
  • Rodrigues AD; Medicine Design-PDM, Worldwide Research and Development, Pfizer Inc., Groton, Connecticut, USA.
  • Temesszentandrási-Ambrus C; SOLVO Biotechnology, a Charles River Company, Budapest, Hungary.
  • Kovács-Hajdu P; SOLVO Biotechnology, a Charles River Company, Budapest, Hungary.
  • Nerada Z; SOLVO Biotechnology, a Charles River Company, Budapest, Hungary.
  • Gáborik Z; SOLVO Biotechnology, a Charles River Company, Budapest, Hungary.
  • Costales C; Medicine Design-PDM, Worldwide Research and Development, Pfizer Inc., Groton, Connecticut, USA. Electronic address: chester.costales@pfizer.com.
J Pharm Sci ; 112(6): 1715-1723, 2023 06.
Article em En | MEDLINE | ID: mdl-36682487

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Tipo de estudo: Etiology_studies / Prognostic_studies / Risk_factors_studies Limite: Animals Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Tipo de estudo: Etiology_studies / Prognostic_studies / Risk_factors_studies Limite: Animals Idioma: En Ano de publicação: 2023 Tipo de documento: Article