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Covalent S-Adenosylhomocysteine-Based DNA Methyltransferase 2 Inhibitors with a New Type of Aryl Warhead.
Schwickert, Marvin; Zimmermann, Robert A; Habeck, Tanja; Hoba, Sabrina N; Nidoieva, Zarina; Fischer, Tim R; Stark, Martin M; Kersten, Christian; Lermyte, Frederik; Helm, Mark; Schirmeister, Tanja.
Afiliação
  • Schwickert M; Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudinger Weg 5, D-55128 Mainz, Germany.
  • Zimmermann RA; Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudinger Weg 5, D-55128 Mainz, Germany.
  • Habeck T; Technical University of Darmstadt, Alarich-Weiss-Strasse 4, D-64287 Darmstadt, Germany.
  • Hoba SN; Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudinger Weg 5, D-55128 Mainz, Germany.
  • Nidoieva Z; Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudinger Weg 5, D-55128 Mainz, Germany.
  • Fischer TR; Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudinger Weg 5, D-55128 Mainz, Germany.
  • Stark MM; Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudinger Weg 5, D-55128 Mainz, Germany.
  • Kersten C; Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudinger Weg 5, D-55128 Mainz, Germany.
  • Lermyte F; Technical University of Darmstadt, Alarich-Weiss-Strasse 4, D-64287 Darmstadt, Germany.
  • Helm M; Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudinger Weg 5, D-55128 Mainz, Germany.
  • Schirmeister T; Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudinger Weg 5, D-55128 Mainz, Germany.
ACS Med Chem Lett ; 14(6): 777-787, 2023 Jun 08.
Article em En | MEDLINE | ID: mdl-37312859

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2023 Tipo de documento: Article