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Tetrazole and oxadiazole derivatives as bioisosteres of tariquidar and elacridar: New potent P-gp modulators acting as MDR reversers.
Braconi, Laura; Dei, Silvia; Contino, Marialessandra; Riganti, Chiara; Bartolucci, Gianluca; Manetti, Dina; Romanelli, Maria Novella; Perrone, Maria Grazia; Colabufo, Nicola Antonio; Guglielmo, Stefano; Teodori, Elisabetta.
Afiliação
  • Braconi L; Department of Neuroscience, Psychology, Drug Research and Child Health - Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Via Ugo Schiff 6, 50019, Sesto Fiorentino, Italy.
  • Dei S; Department of Neuroscience, Psychology, Drug Research and Child Health - Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Via Ugo Schiff 6, 50019, Sesto Fiorentino, Italy. Electronic address: silvia.dei@unifi.it.
  • Contino M; Department of Pharmacy - Drug Sciences, University of Bari "A. Moro", via Orabona 4, 70125, Bari, Italy.
  • Riganti C; Department of Oncology, University of Turin, Via Santena 5/bis, 10126, Torino, Italy.
  • Bartolucci G; Department of Neuroscience, Psychology, Drug Research and Child Health - Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Via Ugo Schiff 6, 50019, Sesto Fiorentino, Italy.
  • Manetti D; Department of Neuroscience, Psychology, Drug Research and Child Health - Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Via Ugo Schiff 6, 50019, Sesto Fiorentino, Italy.
  • Romanelli MN; Department of Neuroscience, Psychology, Drug Research and Child Health - Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Via Ugo Schiff 6, 50019, Sesto Fiorentino, Italy.
  • Perrone MG; Department of Pharmacy - Drug Sciences, University of Bari "A. Moro", via Orabona 4, 70125, Bari, Italy.
  • Colabufo NA; Department of Pharmacy - Drug Sciences, University of Bari "A. Moro", via Orabona 4, 70125, Bari, Italy.
  • Guglielmo S; Department of Drug Science and Technology, University of Turin, Via P. Giuria 9, 10125, Torino, Italy.
  • Teodori E; Department of Neuroscience, Psychology, Drug Research and Child Health - Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Via Ugo Schiff 6, 50019, Sesto Fiorentino, Italy.
Eur J Med Chem ; 259: 115716, 2023 Nov 05.
Article em En | MEDLINE | ID: mdl-37573829

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2023 Tipo de documento: Article