1.
Bioorg Med Chem Lett
; 19(10): 2780-4, 2009 May 15.
Artículo
en Inglés
| MEDLINE
| ID: mdl-19369077
RESUMEN
A series of 4-azaindole inhibitors of c-Met kinase is described. The postulated binding mode was confirmed by an X-ray crystal structure and series optimisation was performed on the basis of this structure. Future directions for series development are discussed.