Detalhe da pesquisa
1.
Anterior cingulate cortex-related functional hyperconnectivity underlies sensory hypersensitivity in Grin2b-mutant mice.
Mol Psychiatry
; 2024 May 04.
Artigo
Inglês
| MEDLINE | ID: mdl-38704508
2.
Inhibition of endocytic uptake of severe acute respiratory syndrome coronavirus 2 and endo-lysosomal acidification by diphenoxylate.
Antimicrob Agents Chemother
; : e0034124, 2024 May 14.
Artigo
Inglês
| MEDLINE | ID: mdl-38742905
3.
PredMS: a random forest model for predicting metabolic stability of drug candidates in human liver microsomes.
Bioinformatics
; 38(2): 364-368, 2022 01 03.
Artigo
Inglês
| MEDLINE | ID: mdl-34515778
4.
Differential effects of two phosphodiesterase 4 inhibitors against lipopolysaccharide-induced neuroinflammation in mice.
BMC Neurosci
; 24(1): 39, 2023 07 31.
Artigo
Inglês
| MEDLINE | ID: mdl-37525115
5.
Discovery of (E)-2-(hydroxyimino)-N-(2 ((4methylpentyl)amino)ethyl)acetamide (KR-27425) as a non-pyridinium oxime reactivator of paraoxon-inhibited acetylcholinesterase.
Bioorg Med Chem Lett
; 96: 129504, 2023 11 15.
Artigo
Inglês
| MEDLINE | ID: mdl-37838342
6.
LightBBB: computational prediction model of blood-brain-barrier penetration based on LightGBM.
Bioinformatics
; 37(8): 1135-1139, 2021 05 23.
Artigo
Inglês
| MEDLINE | ID: mdl-33112379
7.
Anti-neuroinflammatory Effects and Brain Pharmacokinetic Properties of Selonsertib, an Apoptosis signal-regulating Kinase 1 Inhibitor, in mice.
Neurochem Res
; 47(12): 3829-3837, 2022 Dec.
Artigo
Inglês
| MEDLINE | ID: mdl-36309631
8.
Pharmacokinetics of tafamidis, a transthyretin amyloidosis drug, in rats.
Xenobiotica
; 48(8): 831-838, 2018 Aug.
Artigo
Inglês
| MEDLINE | ID: mdl-28803538
9.
Synthesis and Molecular Modeling Studies of N'-Hydroxyindazolecarboximidamides as Novel Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitors.
Molecules
; 22(11)2017 Nov 09.
Artigo
Inglês
| MEDLINE | ID: mdl-29120388
10.
Novel 2,4-diaminopyrimidines bearing tetrahydronaphthalenyl moiety against anaplastic lymphoma kinase (ALK): Synthesis, in vitro, ex vivo, and in vivo efficacy studies.
Bioorg Med Chem Lett
; 26(7): 1720-5, 2016 Apr 01.
Artigo
Inglês
| MEDLINE | ID: mdl-26923695
11.
Discovery of novel tetrahydroisoquinoline-containing pyrimidines as ALK inhibitors.
Bioorg Med Chem
; 24(2): 207-19, 2016 Jan 15.
Artigo
Inglês
| MEDLINE | ID: mdl-26712094
12.
Synthesis and evaluation of novel 2,4-diaminopyrimidines bearing bicyclic aminobenzazepines for anaplastic lymphoma kinase (ALK) inhibitor.
Bioorg Med Chem Lett
; 25(18): 3992-8, 2015 Sep 15.
Artigo
Inglês
| MEDLINE | ID: mdl-26235945
13.
Preclinical pharmacokinetic characterization of 2-(4-(4-(5-(2-phenyl-5-(trifluoromethyl)oxazole-4-carboxamido)-1H-benzo[d]imidazol-2-yl)phenyl)cyclohexyl) acetic acid, a novel DGAT-1 inhibitor.
Xenobiotica
; 44(5): 465-71, 2014 May.
Artigo
Inglês
| MEDLINE | ID: mdl-24152122
14.
PredPS: Attention-based graph neural network for predicting stability of compounds in human plasma.
Comput Struct Biotechnol J
; 21: 3532-3539, 2023.
Artigo
Inglês
| MEDLINE | ID: mdl-37484492
15.
Integrative Analyses Reveal the Anticancer Mechanisms and Sensitivity Markers of the Next-Generation Hypomethylating Agent NTX-301.
Cancers (Basel)
; 15(6)2023 Mar 13.
Artigo
Inglês
| MEDLINE | ID: mdl-36980623
16.
Novel tubulin polymerization inhibitors overcome multidrug resistance and reduce melanoma lung metastasis.
Pharm Res
; 29(11): 3040-52, 2012 Nov.
Artigo
Inglês
| MEDLINE | ID: mdl-22410804
17.
Orally bioavailable tubulin antagonists for paclitaxel-refractory cancer.
Pharm Res
; 29(11): 3053-63, 2012 Nov.
Artigo
Inglês
| MEDLINE | ID: mdl-22760659
18.
Pharmacokinetics and Tissue Distribution of 13C-Labeled Succinic Acid in Mice.
Nutrients
; 14(22)2022 Nov 10.
Artigo
Inglês
| MEDLINE | ID: mdl-36432443
19.
Antibacterial Activity against Clinical Isolates and In Vivo Efficacy of Coralmycins.
Antibiotics (Basel)
; 11(7)2022 Jul 06.
Artigo
Inglês
| MEDLINE | ID: mdl-35884156
20.
Discovery and synthesis of 1,2,4-oxadiazole derivatives as novel inhibitors of Zika, dengue, Japanese encephalitis, and classical swine fever virus infections.
Arch Pharm Res
; 45(4): 280-293, 2022 Apr.
Artigo
Inglês
| MEDLINE | ID: mdl-35441964