Detalhe da pesquisa
1.
Application of a Dual Catalytic Nickel/Iridium-Based Photoredox Reaction to Synthesize 2-Alkyl-N-Arylindoles in a Continuous Flow.
J Org Chem
; 85(19): 12644-12656, 2020 10 02.
Artigo
Inglês
| MEDLINE | ID: mdl-32915566
2.
Visible-Light-Mediated N-Desulfonylation of N-Heterocycles Using a Heteroleptic Copper(I) Complex as a Photocatalyst.
J Org Chem
; 85(13): 8732-8739, 2020 07 02.
Artigo
Inglês
| MEDLINE | ID: mdl-32482067
3.
C-H Functionalization of Heteroarenes Using Unactivated Alkyl Halides through Visible-Light Photoredox Catalysis under Basic Conditions.
J Org Chem
; 83(18): 10933-10940, 2018 09 21.
Artigo
Inglês
| MEDLINE | ID: mdl-30092130
4.
Generation of Diversity Sets with High sp3 Fraction Using the Photoredox Coupling of Organotrifluoroborates and Organosilicates with Heteroaryl/Aryl Bromides in Continuous Flow.
J Org Chem
; 83(3): 1551-1557, 2018 02 02.
Artigo
Inglês
| MEDLINE | ID: mdl-29281285
5.
Application of the Photoredox Coupling of Trifluoroborates and Aryl Bromides to Analog Generation Using Continuous Flow.
J Org Chem
; 81(24): 12525-12531, 2016 12 16.
Artigo
Inglês
| MEDLINE | ID: mdl-27978728
6.
Isosteric replacements of the carboxylic acid of drug candidate VX-787: Effect of charge on antiviral potency and kinase activity of azaindole-based influenza PB2 inhibitors.
Bioorg Med Chem Lett
; 25(9): 1990-4, 2015 May 01.
Artigo
Inglês
| MEDLINE | ID: mdl-25827523
7.
A case of pericardial schistosomiasis and non-Hodgkin high grade B-cell lymphoma.
S Afr J Infect Dis
; 38(1): 524, 2023.
Artigo
Inglês
| MEDLINE | ID: mdl-37795202
8.
A novel series of potent and selective EP(4) receptor ligands: facile modulation of agonism and antagonism.
Bioorg Med Chem Lett
; 21(1): 484-7, 2011 Jan 01.
Artigo
Inglês
| MEDLINE | ID: mdl-21126875
9.
Difluoroethylamines as an amide isostere in inhibitors of cathepsin K.
Bioorg Med Chem Lett
; 21(3): 920-3, 2011 Feb 01.
Artigo
Inglês
| MEDLINE | ID: mdl-21232956
10.
Discovery of Novel, Orally Bioavailable Pyrimidine Ether-Based Inhibitors of ELOVL1.
J Med Chem
; 64(24): 17777-17794, 2021 12 23.
Artigo
Inglês
| MEDLINE | ID: mdl-34871500
11.
Zinc chloride-promoted aryl bromide-alkyne cross-coupling reactions at room temperature.
J Org Chem
; 74(22): 8897-900, 2009 Nov 20.
Artigo
Inglês
| MEDLINE | ID: mdl-19860393
12.
Investigation of ketone warheads as alternatives to the nitrile for preparation of potent and selective cathepsin K inhibitors.
Bioorg Med Chem Lett
; 19(3): 675-9, 2009 Feb 01.
Artigo
Inglês
| MEDLINE | ID: mdl-19117756
13.
Discovery of Novel, Orally Bioavailable ß-Amino Acid Azaindole Inhibitors of Influenza PB2.
ACS Med Chem Lett
; 8(2): 256-260, 2017 Feb 09.
Artigo
Inglês
| MEDLINE | ID: mdl-28197322
14.
Synthesis of Cycloalkyl Substituted 7-Azaindoles via Photoredox Nickel Dual Catalytic Cross-Coupling in Batch and Continuous Flow.
Org Lett
; 18(23): 6180-6183, 2016 12 02.
Artigo
Inglês
| MEDLINE | ID: mdl-27934358
15.
Discovery of a novel, first-in-class, orally bioavailable azaindole inhibitor (VX-787) of influenza PB2.
J Med Chem
; 57(15): 6668-78, 2014 Aug 14.
Artigo
Inglês
| MEDLINE | ID: mdl-25019388