Detalhe da pesquisa
1.
Discovery of NMS-E973 as novel, selective and potent inhibitor of heat shock protein 90 (Hsp90).
Bioorg Med Chem
; 21(22): 7047-63, 2013 Nov 15.
Artigo
Inglês
| MEDLINE | ID: mdl-24100158
2.
NMS-P937, a 4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline derivative as potent and selective Polo-like kinase 1 inhibitor.
Bioorg Med Chem Lett
; 21(10): 2969-74, 2011 May 15.
Artigo
Inglês
| MEDLINE | ID: mdl-21470862
3.
4,5-Dihydro-1H-pyrazolo[4,3-h]quinazolines as potent and selective Polo-like kinase 1 (PLK1) inhibitors.
Bioorg Med Chem Lett
; 20(22): 6489-94, 2010 Nov 15.
Artigo
Inglês
| MEDLINE | ID: mdl-20932759
4.
Catecholic flavonoids acting as telomerase inhibitors.
J Med Chem
; 47(26): 6466-75, 2004 Dec 16.
Artigo
Inglês
| MEDLINE | ID: mdl-15588081
5.
Identification of 4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline derivatives as a new class of orally and selective Polo-like kinase 1 inhibitors.
J Med Chem
; 53(9): 3532-51, 2010 May 13.
Artigo
Inglês
| MEDLINE | ID: mdl-20397705